SCHEMBL29763071

SCHEMBL29763071

FC(F)(F)c1cnc(NC2CCNCC2)nc1O[C@H]1CCOC1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ULK1 O75385 2/20 0.44
FLT3 P36888 2/20 0.42
PTK2 Q05397 4/20 0.41
CHEK1 O14757 2/20 0.41
CDK1 P06493 2/20 0.41
CDK2 P24941 7/20 0.40
KDR P35968 1/20 0.40
MAPK3 P27361 1/20 0.39
MAPK1 P28482 1/20 0.39
CCNK O75909 6/20 0.39
CDK12 Q9NYV4 6/20 0.39
CCNE1 P24864 6/20 0.39
CCNT1 O60563 5/20 0.39
CDK9 P50750 5/20 0.39
CDK7 P50613 2/20 0.38
CCNH P51946 2/20 0.38
MNAT1 P51948 2/20 0.38
CCNB1 P14635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26920117 1.00 ULK1 (0.44) ULK1FLT3PTK2CHEK1CDK1
SCHEMBL26920123 1.00 ULK1 (0.44) ULK1FLT3PTK2CHEK1CDK1
SCHEMBL26943236 0.84 IKBKB (0.47) PTK2CDK1CDK2KDRCCNE1
SCHEMBL26918911 0.82 PTK2 (0.42) ULK1PTK2CDK1CDK2MAPK3
SCHEMBL26918921 0.82 PTK2 (0.42) ULK1PTK2CDK1CDK2MAPK3
SCHEMBL26943136 0.82 IKBKB (0.45) CDK1CDK2KDRCCNE1CCNT1
SCHEMBL25522696 0.81 ULK1 (0.55) ULK1PTK2CDK1CDK2KDR
SCHEMBL26943302 0.80 IKBKB (0.45) CDK1CDK2KDRCCNKCDK12
SCHEMBL31006885 0.80 CCNK (0.56) CDK2CCNKCDK12CCNE1CCNT1
SCHEMBL25531573 0.80 CCNK (0.56) CDK2CCNKCDK12CCNE1CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116472270-A CDK inhibitors 上海齐鲁制药研究中心有限公司 2023-07-21 CN disclosed
WO-2022166793-A1 CDK INHIBITOR 上海齐鲁制药研究中心有限公司 2022-08-11 WO disclosed