SCHEMBL2691981

SCHEMBL2691981

CC(C)OC(=O)O[CH]C1CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.32
OPRK1 P41145 1/20 0.32
CA12 O43570 2/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
MMP2 P08253 2/20 0.32
CA9 Q16790 2/20 0.32
EPHX1 P07099 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9852667 0.80 TSHR (0.34) TSHRCA12CA1CA2MMP2
SCHEMBL4200003 0.77 TSHR (0.38) TSHREPHX1
SCHEMBL2908887 0.77 TSHR (0.36) TSHRCA12CA1CA2MMP2
SCHEMBL698468 0.74 ALDH1A1 (0.43) TSHRNPSR1
SCHEMBL2900646 0.74 CES2 (0.33) TSHREPHX1NPSR1
SCHEMBL2191890 0.73 EPHX1 (0.41) CA12CA1CA2CA9EPHX1
SCHEMBL2905522 0.73 GRIK1 (0.35) MMP2EPHX1
SCHEMBL696980 0.72 ALDH1A1 (0.44) TSHRNPSR1
SCHEMBL2906496 0.71 HCAR2 (0.34) EPHX1HCAR2
SCHEMBL16731836 0.71 EPHX1 (0.44) TSHRCA12CA1CA2MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8168617-B2 Complex pantoic acid ester neopentyl sulfonyl ester cyclization release prodrugs of acamprosate, compositions thereof, and methods of use XENOPORT, INC. (US) 2012-05-01 US disclosed
US-20090076147-A1 COMPLEX PANTOIC ACID ESTER NEOPENTYL SULFONYL ESTER CYCLIZATION RELEASE PRODRUGS OF ACAMPROSATE, COMPOSITIONS THEREOF, AND METHODS OF USE XENOPORT, INC. 2009-03-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090076147-A1 COMPLEX PANTOIC ACID ESTER NEOPENTYL SULFONYL ESTER CYCLIZATION RELEASE PRODRUGS OF ACAMPROSATE, COMPOSITIONS THEREOF, AND METHODS OF USE ADSL, SLC19A1, SLC25A21 TSHR 2112/4885OPRK1 355/4885CA12 1596/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.