Ethiprole

Ethiprole

SCHEMBL27048

CC[S+]([O-])c1c(C#N)nn(-c2c(Cl)cc(C(F)(F)F)cc2Cl)c1N

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 20/20 0.56
GABRD O14764 20/20 0.56
GABRA1 P14867 20/20 0.56
GABRB1 P18505 20/20 0.56
GABRG2 P18507 20/20 0.56
GABRB3 P28472 20/20 0.56
GABRA5 P31644 20/20 0.56
GABRA3 P34903 20/20 0.56
GABRA2 P47869 20/20 0.56
GABRB2 P47870 20/20 0.56
GABRA4 P48169 20/20 0.56
GABRE P78334 20/20 0.56
GABRA6 Q16445 20/20 0.56
GABRG1 Q8N1C3 20/20 0.56
GABRG3 Q99928 20/20 0.56
GABRQ Q9UN88 20/20 0.56
NR1I2 O75469 1/20 0.56
LMNA P02545 1/20 0.56
CYP3A4 P08684 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethiprole SCHEMBL15756765 1.00 GABRP (0.56) GABRPGABRDGABRA1GABRB1GABRG2
Ethiprole SCHEMBL23754762 0.96 GABRP (0.53) GABRPGABRDGABRA1GABRB1GABRG2
Fipronil SCHEMBL727927 0.95 GABRP (0.52) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL14434179 0.95 GABRB3 (0.51) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL14389621 0.92 GABRB3 (0.54) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL18165226 0.90 GABRP (0.57) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL15900786 0.89 GABRP (0.56) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL7673675 0.88 GABRB3 (0.47) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL41972 0.88 GABRP (0.59) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL677248 0.86 GABRP (0.39) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 24522 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122036637-A Polymorphs 先正达农作物保护股份公司 2026-05-15 CN claimed
EP-4734762-A1 BAIT COMPOSITIONS FMC Corporation (US) 2026-05-06 EP claimed
EP-4719059-A1 INCREASED PALATABILITY OF INSECTICIDAL INSECT BAITS Bio Logic Crop Science, S.L. (ES) 2026-04-08 EP claimed
US-20260083129-A1 PYRAZOLE AMIDE INSECTICIDES FMC CORP (US) 2026-03-26 US claimed
US-20260083130-A1 NOVEL SULFONATE BENZAMIDE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS FMC CORP (US) 2026-03-26 US claimed
EP-4709166-A1 NOVEL INSECTICIDAL MIXTURES FOR CONTROLLING AND PROTECTING CROPS ADAMA MAKHTESHIM LTD. (IL) 2026-03-18 EP claimed
EP-4710766-A1 MIXTURES OF AMBRUTICIN WITH AT LEAST ONE FURTHER PESTICIDE BASF SE (DE) 2026-03-18 EP claimed
US-12568969-B2 Pyridine compounds for controlling invertebrate pests FMC CORPORATION (US) 2026-03-10 US claimed
CN-121577800-A Non-targeted screening multi-pesticide residue detection method based on high-resolution mass spectrum 常州市食品药品纤维质量监督检验中心(常州市粮油质量监督检测站、常州纤维检验所) 2026-02-27 CN claimed
CN-121577795-A Method and system for rapidly determining ethiprole enantiomer residue in tomatoes by solid phase extraction-ultra-high performance synthetic phase chromatography 杭州海关技术中心 2026-02-27 CN claimed
EP-1165485-A2 PROCESSES FOR PREPARING PESTICIDAL INTERMEDIATES AVENTIS CROPSCIENCE S.A. (FR) 2002-01-02 EP claimed
WO-2001019189-A1 COMPOSITIONS AND METHODS FOR CONTROLLING INSECTS WHICH DAMAGE RICE AND OTHER CROPS AVENTIS CROPSCIENCE S.A. (FR) 2001-03-22 WO claimed
WO-2000059862-A2 PROCESSES FOR PREPARING PESTICIDAL INTERMEDIATES AVENTIS CROPSCIENCE S.A. (FR) 2000-10-12 WO claimed
US-H1900-H APPLYING AN ARYLPYRAZOLES OVICIDE TO THE EGGS OF THE INSECTS RHONE-POULENC AG COMPANY INC. (US) 2000-10-03 US claimed
US-6090751-A AN INSECTICIDAL 1-ARYLPYRAZOLE AND TO PREVENT LARGE CRYSTALS FROM PRECIPITATING: AN N-ALKYLPYRROLIDINONE SOLVENT, A CO-SOLVENT WITH SPECIFIC WATER SOLUBILITY, AND AN EMULSIFIER RHONE-POULENC AGRO (FR) 2000-07-18 US claimed
US-6057355-A SYNERGISTIC MIXTURE OF 1-(4-(2,4-DICHLOROPHENOXY)-2,5-DIMETHYL-3-CHLOROPHENYL)-3-(2,6 -DIFLUOROBEN ZOYL)UREA AND 5-AMINO-3-CYANO-1-(2,6-DICHLORO-4-TRIFLUOROMETHYLPHENYL)-4-TRI RHONE-POULENC INC. (US) 2000-05-02 US claimed
EP-0806895-B1 INSECTICIDAL COMBINATIONS INCLUDING AN INSECTICIDE FROM THE CHLORONICOTINYL FAMILY AND AN INSECTICIDE HAVING A PYRAZOLE, PYRROLE OR PHENYLIMIDAZOLE GROUP RHONE POULENC AGROCHIMIE (FR) 2000-04-12 EP claimed
US-5883112-A INSECTICIDES RHONE-POULENC INC. (US) 1999-03-16 US claimed
US-5814652-A SYSTEMIC INSECTICIDES RHONE-POULENC INC. (US) 1998-09-29 US claimed
WO-1997022593-A1 NOVEL 5-AMINO-3-CYANO-4-ETHYLSULFINYL-1-PHENYL-PYRAZOLE COMPOUNDS AND THEIR USE AS PESTICIDES RHONE-POULENC AGROCHIMIE (FR) 1997-06-26 WO claimed