SCHEMBL2711084

SCHEMBL2711084

Cc1csc(CNC(=O)c2ccccc2)n1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.58
RAB9A P51151 4/20 0.58
KDM4E B2RXH2 2/20 0.53
HSP90AA1 P07900 1/20 0.53
NAMPT P43490 1/20 0.53
MAPT P10636 3/20 0.52
HPGD P15428 4/20 0.51
ALDH1A1 P00352 1/20 0.51
HTT P42858 1/20 0.51
SCD O00767 1/20 0.49
HSD17B10 Q99714 1/20 0.48
LMNA P02545 2/20 0.46
POLB P06746 1/20 0.46
MAPK1 P28482 1/20 0.46
SLC5A7 Q9GZV3 1/20 0.46
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL166396 0.88 NAMPT (0.48) NPC1RAB9AKDM4EHSP90AA1NAMPT
SCHEMBL3507210 0.85 RAB9A (0.51) NPC1RAB9AKDM4EHSP90AA1NAMPT
SCHEMBL3641653 0.84 NAMPT (0.48) NPC1RAB9AKDM4EHSP90AA1NAMPT
SCHEMBL3647405 0.84 ENPP2 (0.52) NPC1RAB9AKDM4EHSP90AA1NAMPT
SCHEMBL2711947 0.83 HPGD (0.56) NPC1RAB9AKDM4EHSP90AA1NAMPT
SCHEMBL7984987 0.82 KDM4E (0.53) NPC1KDM4EMAPTHPGDALDH1A1
SCHEMBL166267 0.82 NAMPT (0.46) NPC1RAB9AKDM4EHSP90AA1NAMPT
SCHEMBL30614797 0.82 ADORA2A (0.54) NPC1RAB9AHSP90AA1NAMPTALDH1A1
SCHEMBL2227256 0.81 MAPT (0.67) NPC1RAB9AKDM4EMAPTHPGD
SCHEMBL7260803 0.80 RAB9A (0.67) NPC1RAB9AKDM4EHSP90AA1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed