SCHEMBL2714906

SCHEMBL2714906

C#Cc1cc(NC(=O)O)ccc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.43
NPC1 O15118 5/20 0.42
RAB9A P51151 5/20 0.42
AKT1 P31749 1/20 0.42
KMT2A Q03164 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
MEN1 O00255 2/20 0.40
LMNA P02545 2/20 0.40
HTT P42858 2/20 0.40
SLC2A1 P11166 1/20 0.39
EGFR P00533 1/20 0.38
FBP1 P09467 1/20 0.38
TSHR P16473 1/20 0.37
MAPT P10636 1/20 0.37
TP53 P04637 1/20 0.37
BLM P54132 1/20 0.36
WRN Q14191 1/20 0.36
TDO2 P48775 1/20 0.36
FABP4 P15090 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4900667 0.83 GRM4 (0.59) GRM4NPC1RAB9AAKT1BLM
SCHEMBL13400510 0.81 MEN1 (0.49) GRM4NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL16088607 0.79 CYP1A2 (0.55) GRM4NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL2092311 0.77 RAB9A (0.65) NPC1RAB9AKMT2ASMN1; SMN2MEN1
SCHEMBL13022995 0.77 NPC1 (0.46) GRM4NPC1RAB9AKMT2AMEN1
SCHEMBL18323173 0.77 NPC1 (0.49) GRM4NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL15907212 0.75 GRM4 (0.39) GRM4NPC1RAB9AAKT1KMT2A
SCHEMBL18323190 0.75 ALDH1A1 (0.53) NPC1RAB9AKMT2ASMN1; SMN2MEN1
SCHEMBL28293553 0.74 EGFR (0.41) GRM4AKT1KMT2AMEN1HTT
SCHEMBL31591018 0.73 LMNA (0.44) RAB9AKMT2ASMN1; SMN2MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012052451-A1 METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2012-04-26 WO disclosed