SCHEMBL28293553

SCHEMBL28293553

C#Cc1cc(NCl)ccc1F

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.41
FBP1 P09467 1/20 0.41
TDO2 P48775 2/20 0.36
GRM4 Q14833 1/20 0.34
AKT1 P31749 1/20 0.33
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2714906 0.74 GRM4 (0.43) EGFRFBP1TDO2GRM4AKT1
SCHEMBL1544963 0.74 PTGDR2 (0.36) EGFRFBP1ALDH1A1KMT2ATSHR
SCHEMBL9844844 0.73 RAPGEF4 (0.45) MEN1ALDH1A1MAPTHTTKMT2A
SCHEMBL718612 0.72 CA3 (0.42) EGFRFBP1ALDH1A1
SCHEMBL17787791 0.68 EGFR (0.32) EGFRFBP1
SCHEMBL2897973 0.68 NFE2L2 (0.36) EGFRFBP1ALDH1A1
SCHEMBL2809900 0.68 ESR1 (0.45)
SCHEMBL19294196 0.68 RAPGEF4 (0.42) TDO2GRM4MEN1ALDH1A1MAPT
SCHEMBL2812282 0.68 TRPV4 (0.47) EGFRFBP1
SCHEMBL5958536 0.68 PYCR1 (0.39) EGFRFBP1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109790122-A Heterocyclic compound 武田药品工业株式会社 2019-05-21 CN disclosed