SCHEMBL27200524

SCHEMBL27200524

NS(=O)(=O)c1ccc(N2CCN(C(=O)O)CC2)c(F)c1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 7/20 0.54
CA2 P00918 11/20 0.46
CA1 P00915 9/20 0.46
CA7 P43166 5/20 0.46
CA9 Q16790 6/20 0.46
CA12 O43570 4/20 0.46
CA14 Q9ULX7 3/20 0.46
ALDH1A1 P00352 1/20 0.45
GPR55 Q9Y2T6 1/20 0.44
CA4 P22748 1/20 0.44
CA6 P23280 1/20 0.44
CA5A P35218 1/20 0.44
CA5B Q9Y2D0 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20502378 0.81 CA2 (0.59) SLC6A9CA2CA1CA7CA9
SCHEMBL3922259 0.80 MAPT (0.63) SLC6A9ALDH1A1GPR55
SCHEMBL632171 0.79 GRM5 (0.59) ALDH1A1
SCHEMBL5037826 0.79 SLC6A9 (0.71) SLC6A9GPR55
SCHEMBL20502523 0.78 ALDH1A1 (0.53) CA2CA1CA7CA9CA12
SCHEMBL3923062 0.78 ALDH1A1 (0.58) SLC6A9CA2CA1CA7CA9
SCHEMBL4133081 0.78 GRM5 (0.48) ALDH1A1
SCHEMBL3930029 0.78 SLC6A9 (0.88) SLC6A9GPR55
SCHEMBL20141519 0.78 CA12 (0.46) CA2CA1CA7CA9CA12
SCHEMBL19212228 0.77 ALDH1A1 (0.58) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3596059-B1 HETEROCYCLIC COMPOUNDS USEFUL AS DUAL ATX/CA INHIBITORS HOFFMANN LA ROCHE (CH) 2024-04-24 EP claimed
CN-110392679-B Heterocyclic compounds useful as dual ATX/CA inhibitors 豪夫迈·罗氏有限公司 2023-04-07 CN disclosed