SCHEMBL2721044

SCHEMBL2721044

O=C(Cl)c1c(Cl)sc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.49
HDAC1 Q13547 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
LMNA P02545 1/20 0.45
MAPK1 P28482 1/20 0.45
OGG1 O15527 1/20 0.44
GPR3 P46089 1/20 0.43
ALDH1A1 P00352 2/20 0.42
IKBKB O14920 1/20 0.41
LIMK1 P53667 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRA5 P31644 1/20 0.41
CD274 Q9NZQ7 1/20 0.41
ACLY P53396 1/20 0.40
KDM4E B2RXH2 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
LOXL2 Q9Y4K0 1/20 0.39
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8666781 0.85 MCL1 (0.58) MCL1HDAC1HDAC8HDAC6LMNA
SCHEMBL27629193 0.81 MCL1 (0.53) MCL1HDAC1HDAC8HDAC6LMNA
SCHEMBL3192118 0.79 LMNA (0.69) MCL1HDAC1HDAC8HDAC6LMNA
SCHEMBL15700018 0.75 LMNA (0.41) MCL1HDAC1HDAC8HDAC6LMNA
SCHEMBL64428 0.73 MCL1 (0.73) MCL1HDAC1HDAC8HDAC6LMNA
SCHEMBL30368759 0.71 ALDH1A1 (0.52) ALDH1A1KDM4EALOX15
SCHEMBL11674250 0.71 ALDH1A1 (0.52) ALDH1A1KDM4EALOX15
SCHEMBL28540289 0.71 GPR3 (0.50) MCL1HDAC1HDAC8HDAC6LMNA
SCHEMBL28322189 0.70 LOXL2 (0.57) MCL1HDAC1HDAC8HDAC6LMNA
SCHEMBL15557963 0.69 ALDH1A1 (0.50) MCL1LMNAALDH1A1KDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2635559-A2 NEUROTRYPSIN INHIBITORS Neurotune AG (CH) 2013-09-11 EP disclosed
WO-2012059442-A2 NEUROTRYPSIN INHIBITORS NEUROTUNE AG (CH) 2012-05-10 WO disclosed