SCHEMBL2722140

SCHEMBL2722140

COc1ccc(C2CC2C(=O)O)cc1I

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.50
SLC6A4 P31645 1/20 0.50
SLC6A3 Q01959 1/20 0.50
APP P05067 2/20 0.46
FFAR1 O14842 3/20 0.45
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA9 Q16790 2/20 0.45
CA12 O43570 1/20 0.45
RXRA P19793 1/20 0.44
LTB4R Q15722 1/20 0.43
PDE4B Q07343 2/20 0.42
MAPT P10636 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PDE4A P27815 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
TRPM5 Q9NZQ8 2/20 0.41
TUBB4A P04350 3/20 0.40
TUBB P07437 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2722142 1.00 SLC6A2 (0.50) SLC6A2SLC6A4SLC6A3APPFFAR1
SCHEMBL7002288 0.86 APP (0.55) SLC6A2SLC6A4SLC6A3APPFFAR1
SCHEMBL7002284 0.86 APP (0.55) SLC6A2SLC6A4SLC6A3APPFFAR1
SCHEMBL2952559 0.86 APP (0.55) SLC6A2SLC6A4SLC6A3APPFFAR1
SCHEMBL7002924 0.84 RXRA (0.49) APPFFAR1CA1CA2CA9
SCHEMBL10254282 0.84 RXRA (0.49) APPFFAR1CA1CA2CA9
SCHEMBL6996736 0.82 ALDH1A1 (0.52) APPFFAR1CA1CA2CA9
SCHEMBL7000989 0.82 KDM1A (0.61) SLC6A2SLC6A4SLC6A3APPFFAR1
SCHEMBL6996735 0.82 ALDH1A1 (0.52) APPFFAR1CA1CA2CA9
SCHEMBL15669063 0.82 KDM1A (0.61) SLC6A2SLC6A4SLC6A3APPFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632269-A1 CYCLIC AMINE SUBSTITUTED OXAZOLIDINONE CETP INHIBITOR Merck Sharp & Dohme Corp. (US) 2013-09-04 EP disclosed
WO-2012058187-A1 CYCLIC AMINE SUBSTITUTED OXAZOLIDINONE CETP INHIBITOR MERCK SHARP & DOHME CORP. (US) 2012-05-03 WO disclosed