SCHEMBL2728147

SCHEMBL2728147

Cc1csc([C@H]2CCCN2C(=O)c2cc(-c3nnc([C@@](C)(Cc4ccccc4)NC(=O)O)o3)nc(-n3ccnc3)c2)n1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.34
NAPEPLD Q6IQ20 1/20 0.34
NOS2 P35228 5/20 0.34
NOS1 P29475 3/20 0.34
TRPV1 Q8NER1 3/20 0.34
ROCK2 O75116 3/20 0.33
POLB P06746 1/20 0.32
CPT2 P23786 2/20 0.32
CPT1A P50416 2/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
PKM P14618 1/20 0.31
CD38 P28907 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6467759 0.95 SMN1; SMN2 (0.34) SMN1; SMN2NAPEPLDNOS2NOS1TRPV1
SCHEMBL2726650 0.92 NAPEPLD (0.34) NAPEPLDNOS2NOS1TRPV1ROCK2
SCHEMBL2726646 0.92 NAPEPLD (0.34) NAPEPLDNOS2NOS1TRPV1ROCK2
SCHEMBL2728180 0.90 HCRTR1 (0.38) SMN1; SMN2TRPV1POLBHCRTR1HCRTR2
SCHEMBL2728191 0.90 SMN1; SMN2 (0.38) SMN1; SMN2TRPV1POLBCPT2CPT1A
SCHEMBL2728838 0.90 ROCK2 (0.34) SMN1; SMN2NAPEPLDNOS2NOS1TRPV1
SCHEMBL2727446 0.89 SMN1; SMN2 (0.35) SMN1; SMN2NAPEPLDTRPV1POLBHCRTR1
SCHEMBL2727845 0.89 CPT1A (0.39) SMN1; SMN2TRPV1POLBCPT2CPT1A
Fumaric Acid SCHEMBL2733545 0.89 NAPEPLD (0.33) NAPEPLDNOS2NOS1TRPV1ROCK2
SCHEMBL2725371 0.89 SMN1; SMN2 (0.34) SMN1; SMN2TRPV1POLBCPT2CPT1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed