SCHEMBL27314830

SCHEMBL27314830

CC(C)(F)c1cncc(O)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.39
GABRB2 P47870 1/20 0.39
APLNR P35414 1/20 0.35
HSD17B1 P14061 1/20 0.32
CYP11B2 P19099 7/20 0.32
CYP11B1 P15538 5/20 0.32
HPGD P15428 2/20 0.31
HSD17B10 Q99714 2/20 0.31
ALDH1A1 P00352 1/20 0.31
ALOX15 P16050 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
POLB P06746 2/20 0.31
ESR2 Q92731 2/20 0.31
RECQL P46063 1/20 0.31
CHRNB2 P17787 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
CHRNA4 P43681 1/20 0.30
CYP19A1 P11511 2/20 0.30
CYP2C9 P11712 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27314463 0.87 GABRA1 (0.39) GABRA1GABRB2APLNRHSD17B1CYP11B2
SCHEMBL8170002 0.82 GABRA1 (0.54) GABRA1GABRB2APLNRHSD17B1CYP11B2
SCHEMBL875313 0.82 TAS2R14 (0.38) APLNRCYP11B2CYP11B1ALDH1A1CYP19A1
SCHEMBL13885073 0.78 APLNR (0.35) GABRA1GABRB2APLNRHSD17B1POLB
SCHEMBL19366826 0.77 GABRA1 (0.37) GABRA1GABRB2POLBKDM4EGAA
SCHEMBL24680657 0.76 HCAR2 (0.38) CYP11B2CYP11B1CYP19A1AR
SCHEMBL30879971 0.76 HCAR2 (0.38) CYP11B2CYP11B1CYP19A1AR
SCHEMBL21958802 0.76 HCAR2 (0.38) CYP11B2CYP11B1CYP19A1CYP2C9CYP3A4
SCHEMBL20458840 0.75 GABRA1 (0.37) GABRA1GABRB2APLNRHSD17B1POLB
SCHEMBL24534066 0.74 KDM4E (0.36) CYP11B2CYP11B1ALDH1A1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024091542-A1 COMPOUNDS AND COMPOSITIONS AS GPR52 MODULATORS NEUROCRINE BIOSCIENCES, INC. (US) 2024-05-02 WO disclosed
WO-2024091542-A1 COMPOUNDS AND COMPOSITIONS AS GPR52 MODULATORS NEUROCRINE BIOSCIENCES, INC. (US) 2024-05-02 WO disclosed