SCHEMBL2732828

SCHEMBL2732828

Brc1cccc(-c2cc(-c3cccnc3)no2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.50
CYP2C19 P33261 5/20 0.50
CYP2A6 P11509 2/20 0.50
CYP2E1 P05181 1/20 0.50
CYP2B6 P20813 1/20 0.50
CYP1A2 P05177 5/20 0.46
CYP3A4 P08684 5/20 0.46
CYP2D6 P10635 3/20 0.46
CHRNB2 P17787 2/20 0.45
CHRNA5 P30532 2/20 0.45
CHRNA4 P43681 2/20 0.45
NPC1 O15118 5/20 0.45
RAB9A P51151 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
TP53 P04637 2/20 0.45
PKM P14618 2/20 0.45
TSHR P16473 1/20 0.45
CA9 Q16790 1/20 0.43
CYP19A1 P11511 3/20 0.43
HSD17B10 Q99714 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15293831 0.84 CYP2A6 (0.68) CYP2C9CYP2C19CYP2A6CYP2E1CYP2B6
SCHEMBL2017685 0.83 CYP2A6 (0.62) CYP2A6CYP1A2CYP3A4SMN1; SMN2TP53
SCHEMBL4318440 0.81 CYP3A4 (0.62) CYP2C9CYP2C19CYP2A6CYP2E1CYP2B6
SCHEMBL23843626 0.79 CYP19A1 (0.60) CYP2A6CYP1A2CYP3A4CYP19A1ALDH1A1
SCHEMBL4322525 0.79 RAB9A (0.70) CYP2C9CYP2C19CYP2A6CYP2E1CYP2B6
SCHEMBL15293840 0.78 NPC1 (0.53) CYP2C9CYP2C19CYP2A6CYP2E1CYP2B6
SCHEMBL4316802 0.78 MAPT (0.59) CYP2C9CYP2C19CYP2A6CYP2E1CYP2B6
SCHEMBL2462787 0.77 CHRNB2 (0.69) CHRNB2CHRNA5CHRNA4NPC1RAB9A
SCHEMBL15293856 0.76 NPC1 (0.60) CYP2C9CYP2C19CYP2A6CYP2E1CYP2B6
SCHEMBL4325908 0.75 CYP2C9 (0.65) CYP2C9CYP2C19CYP2A6CYP2E1CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150373978-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER IP GMBH (DE) 2015-12-31 US disclosed
US-20150373978-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER IP GMBH (DE) 2015-12-31 US disclosed
US-20150373978-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER IP GMBH (DE) 2015-12-31 US disclosed
US-9173396-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-11-03 US disclosed
US-9173396-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-11-03 US disclosed
US-9173396-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-11-03 US disclosed
US-20130261141-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-10-03 US disclosed
US-20130261141-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-10-03 US disclosed
US-20130261141-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-10-03 US disclosed
EP-2630133-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES Bayer Intellectual Property GmbH (DE) 2013-08-28 EP disclosed
WO-2012052412-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2012-04-26 WO disclosed
WO-2012052412-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2012-04-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130261141-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES DDT, ACHE, PTMS CYP2C9 337/4885CYP2C19 1286/4885CYP2A6 853/4885
US-20150373978-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES DDT, ACHE, PTMS CYP2C9 337/4885CYP2C19 1286/4885CYP2A6 853/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.