SCHEMBL27337277

SCHEMBL27337277

NC(=O)NSc1cccc(F)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.49
PARP1 P09874 1/20 0.47
KCNN4 O15554 4/20 0.43
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
TSHR P16473 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NR3C2 P08235 1/20 0.38
HAO1 Q9UJM8 1/20 0.38
IKBKB O14920 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28248610 0.82 EPHX1 (0.42) EPHX1PARP1KCNN4CES2CES1
SCHEMBL27687143 0.80 PARP1 (0.46) PARP1MEN1KMT2AIKBKB
SCHEMBL27301554 0.79 PARP1 (0.47) PARP1MEN1KMT2AIKBKB
SCHEMBL27605662 0.79 PARP1 (0.47) PARP1HDAC6MEN1KMT2ANR3C2
SCHEMBL27608065 0.79 PARP1 (0.47) PARP1MEN1KMT2A
SCHEMBL27928000 0.79 CYP1A2 (0.35) HDAC1
SCHEMBL27708208 0.78 KDM4E (0.59) EPHX1CES2MEN1KMT2A
SCHEMBL27639755 0.77 PRSS1 (0.44) IKBKB
SCHEMBL27317150 0.77 ALDH1A1 (0.50) KCNN4CES2CES1HDAC6MEN1
SCHEMBL158241 0.77 SIRT1 (0.42) PARP1TSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101687816-A Triaminopyrimidine derivatives as the CDC25 inhibitors of phosphatases IPSEN PHARMA SAS 2010-03-31 CN claimed
CN-108137528-A Pleocidin derivative as insecticide 阿格里麦蒂斯有限责任公司 2018-06-08 CN disclosed
CN-107235916-A A kind of licochalcone A deracil analog derivative and its synthetic method for having antitumor activity 陕西科技大学 2017-10-10 CN disclosed
CN-104540835-B The imidazo thiadiazoles derivative as proteinase activated receptors 4 (PAR4) inhibitor for treating platelet aggregation 百时美施贵宝公司 2017-08-08 CN disclosed
CN-103476764-B Process for producing episulfide compound ASAHI KASEI KABUSHIKI KAISHA (JP) 2016-05-25 CN disclosed
CN-103288721-B (4-(4-[6-(trifluoromethylpyridin-3-base amino)-containing N heteroaryl]-phenyl)-cyclohexyl)-acetogenin and pharmaceutical use thereof NOVARTIS AG (CH) 2016-04-20 CN disclosed
CN-104610222-A Process for preparing episulfide compounds ASAHI KASEI CHEMICALS CORP 2015-05-13 CN disclosed
CN-104540835-A Imidazothiadiazole derivatives as protease activated receptor 4 (par4) inhibitors for treating platelet aggregation BRISTOL MYERS SQUIBB CO 2015-04-22 CN disclosed
CN-103476764-A Process for producing episulfide compound ASAHI KASEI CHEMICALS CORP (JP) 2013-12-25 CN disclosed
CN-103288721-A (4-(4-[6-(trifluoromethyl-pyridin-3-ylamino)-n-containing-heteroaryl]-phenyl)-cyclohexyl)-acetic acid derivatives and pharmaceutical uses thereof NOVARTIS AG 2013-09-11 CN disclosed
CN-101415683-B Novel compounds NOVARTIS AG 2013-07-17 CN disclosed
CN-103086981-A New compounds NOVARTIS AG 2013-05-08 CN disclosed
CN-102367240-A 1,2,3-thiadiazole mother ring-contained iminothiazolone compounds, intermediate thereof, and preparation methods and applications of compound and intermediate UNIV EAST CHINA SCIENCE & TECH 2012-03-07 CN disclosed
CN-101687816-A Triaminopyrimidine derivatives as the CDC25 inhibitors of phosphatases IPSEN PHARMA SAS 2010-03-31 CN disclosed
CN-101415683-A Novel compounds NOVARTIS AG (CH) 2009-04-22 CN disclosed
CN-1043891-C Fluorobenzothiazolyloxyacetamides BAYER AG (DE) 1999-06-30 CN disclosed
CN-1087903-A Fluoro benzothiazole oxygen yl acetamide BAYER AG (DE) 1994-06-15 CN disclosed