SCHEMBL158241

SCHEMBL158241

NC(=O)NSc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 2/20 0.42
MAPT P10636 3/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 2/20 0.41
HSD17B10 Q99714 2/20 0.41
POLB P06746 1/20 0.41
PARP1 P09874 1/20 0.41
TSHR P16473 1/20 0.41
RECQL P46063 1/20 0.41
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
GAA P10253 2/20 0.41
GFER P55789 1/20 0.41
FFAR1 O14842 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
ALDH1A1 P00352 4/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethylamine SCHEMBL27576834 0.94 LMNA (0.40) SIRT1MAPTCYP3A4CYP2C19HSD17B10
SCHEMBL6034931 0.90 MTNR1A (0.42) SIRT1MAPTCYP3A4CYP2C19HSD17B10
SCHEMBL4558245 0.88 NPC1 (0.41) MAPTTSHRGAALMNANPC1
Propanol SCHEMBL28703544 0.87 MTNR1A (0.37) SIRT1CYP3A4CYP2C19FFAR1CYP1A2
SCHEMBL3070802 0.86 FFAR1 (0.43) SIRT1MAPTCYP3A4CYP2C19HSD17B10
SCHEMBL3083062 0.84 POLB (0.43) SIRT1MAPTCYP3A4CYP2C19HSD17B10
SCHEMBL27639739 0.83 PARP10 (0.53) TSHRFFAR1ALDH1A1KMT2AHPGD
SCHEMBL28233528 0.83 TRPA1 (0.47) MAPTPOLBTDP1L3MBTL1CYP1A2
SCHEMBL5528839 0.83 TRPA1 (0.47) MAPTPOLBTDP1L3MBTL1CYP1A2
SCHEMBL27639755 0.83 PRSS1 (0.44) SIRT1MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 827 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025024478-A1 COMPOSITIONS FOR THE MODULATION OF TASTE IXORA SCIENTIFIC INC. (US) 2025-01-30 WO claimed
US-20240410893-A1 COMPOSITIONS, SYSTEMS, AND METHODS FOR DETERMINATION OF T2R AND/OR T1R PHENOTYPE IN INDIVIDUALS TO PREDICT CANNABIS TASTING PREFERENCES, CHARACTERIZATION OF CANNABIS IN RELATION TO INDIVIDUAL TASTING PREFERENCES, AND SELECTION OF CANNABIS Phenomune, LLC (US) 2024-12-12 US claimed
US-20240344126-A1 COMPOSITIONS, SYSTEMS, AND METHODS FOR DETERMINATION OF T2R AND/OR T1R PHENOTYPE IN INDIVIDUALS TO PREDICT WINE TASTING PREFERENCES, CHARACTERIZATION OF WINE IN RELATION TO INDIVIDUAL TASTING PREFERENCES, AND SELECTION OF WINE Phenomune, LLC (US) 2024-10-17 US claimed
US-20240218444-A1 COMPOSITIONS, SYSTEMS, AND METHODS FOR DETERMINATION OF T2R AND/OR T1R PHENOTYPE IN INDIVIDUALS TO PREDICT DISTILLED SPIRIT TASTING PREFERENCES, CHARACTERIZATION OF DISTILLED SPIRIT IN RELATION TO INDIVIDUAL TASTING PREFERENCES, AND SELECTION OF DISTILLED SPIRIT Phenomune, LLC (US) 2024-07-04 US claimed
US-20230184746-A1 HIGH-SENSITIVITY DETECTION OF GPCR ACTIVITY AND USES THEREOF FIRMENICH INCORPORATED 2023-06-15 US claimed
US-20230144186-A1 QUININE AND ITS USE TO GENERATE INNATE IMMUNE RESPONSE THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2023-05-11 US claimed
WO-2023063994-A1 TESTING METHODS FOR DETERMINATION OF T2R PHENOTYPE AND APPLICATIONS THEREOF Phenomune, LLC (US) 2023-04-20 WO claimed
EP-4138835-A1 QUININE AND ITS USE TO GENERATE INNATE IMMUNE RESPONSE Cohen, Noam (US) 2023-03-01 EP claimed
US-20220196654-A1 TESTING METHODS FOR DETERMINATION OF T2R PHENOTYPE AND APPLICATIONS THEREOF Phenomune, LLC (US) 2022-06-23 US claimed
US-20210404068-A1 ETCHING SOLUTION, ANNEXING AGENT, AND MANUFACTURING METHOD OF METAL WIRING TCL CHINA STAR OPTOELECTRONICS TECHNOLOGY CO., LTD. (CN) 2021-12-30 US claimed
US-20030075073-A1 Furniture polish composition S.C. JOHNSON & SON, INC. 2003-04-24 US claimed
US-6383778-B1 NUCLEOTIDE SEQUENCE WHICH CODES FOR RECEPTOR THAT BINDS TO PHENYLTHIOCARBAMIDE LIGAND; FOR TASTE MODULATING COMPOUNDS FOR USE IN FOOD AND DRUG INDUSTRIES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2002-05-07 US claimed
US-6337080-B1 DEVICE FOR DISPENSING AN INSECT CONTROL ACTIVE FORMULATION FOR USE WITH A HEATER FOR THE CONTROL OF INSECTS AND TREATED TO DISCOURAGE INGESTION BY PETS OR MISUSE BY CHILDREN OR OTHER PERSONS S. C. JOHNSON & SON, INC. 2002-01-08 US claimed
WO-2001045506-A1 INSECT CONTROL MAT S. C. JOHNSON & SON, INC. (US) 2001-06-28 WO claimed
EP-0549752-A1 PROTEIN SEQUENCING BECKMAN INSTRUMENTS, INC. (US) 1993-07-07 EP claimed
WO-1993000355-A1 PROTEIN SEQUENCING PORTON INSTRUMENTS, INC. (US) 1993-01-07 WO claimed
EP-0207416-B1 PROCESS FOR THE PREPARATION OF 2-AMINOBENZOTHIAZOLES HOECHST AKTIENGESELLSCHAFT (DE) 1989-08-16 EP claimed
EP-0102055-B1 PROCESS FOR THE PREPARATION OF HALOGEN-SUBSTITUTED 2-AMINO-BENZOTHIAZOLES HOECHST AKTIENGESELLSCHAFT (DE) 1988-05-11 EP claimed
EP-0006587-B1 SULFONYL UREAS, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1981-11-11 EP claimed
EP-0005276-B1 METHOD OF PREPARING MONOARYLTHIOUREA HOECHST AKTIENGESELLSCHAFT (DE) 1981-01-07 EP claimed