SCHEMBL27348192

SCHEMBL27348192

N#Cc1c(CF)cc(Cl)nc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
ALDH1A1 P00352 3/20 0.34
HTT P42858 3/20 0.33
GLA P06280 1/20 0.33
NSD2 O96028 1/20 0.33
MAPK1 P28482 1/20 0.33
KDM1A O60341 4/20 0.32
KDM4E B2RXH2 2/20 0.32
POLB P06746 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31
PPARG P37231 1/20 0.31
NCOA2 Q15596 1/20 0.31
NCOA1 Q15788 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22980966 0.82 KHK (0.34) KHKL3MBTL1ALDH1A1HTTGLA
SCHEMBL11723001 0.81 HTT (0.42) L3MBTL1ALDH1A1HTTGLAMAPK1
SCHEMBL6627580 0.79 ALDH1A1 (0.40) L3MBTL1ALDH1A1HTTGLAMAPK1
SCHEMBL4068543 0.79 L3MBTL1 (0.33) KHKL3MBTL1ALDH1A1HTTGLA
SCHEMBL4193505 0.78 HTT (0.38) KHKL3MBTL1ALDH1A1HTTGLA
SCHEMBL1624060 0.77 L3MBTL1 (0.33) KHKL3MBTL1ALDH1A1HTTGLA
SCHEMBL9987538 0.77 L3MBTL1 (0.33) KHKL3MBTL1ALDH1A1HTTGLA
SCHEMBL21154750 0.75 TAAR1 (0.38) L3MBTL1ALDH1A1HTTGLAKDM4E
SCHEMBL7600961 0.75 TRPV4 (0.43) KHKL3MBTL1ALDH1A1HTTGLA
SCHEMBL30402943 0.74 L3MBTL1 (0.40) KHKL3MBTL1ALDH1A1HTTGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4630114-A1 NEW CYANOPYRIDINE KHK INHIBITOR COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2025-10-15 EP disclosed
WO-2024121183-A1 NEW CYANOPYRIDINE KHK INHIBITOR COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2024-06-13 WO disclosed
WO-2024121183-A1 NEW CYANOPYRIDINE KHK INHIBITOR COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2024-06-13 WO disclosed