SCHEMBL27353158

SCHEMBL27353158

Cc1ncc(-c2ccnn2-c2ccccc2)cn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 1/20 0.50
NR3C2 P08235 3/20 0.46
POLB P06746 1/20 0.44
MAPK9 P45984 2/20 0.44
MAPK10 P53779 2/20 0.44
MAPK8 P45983 1/20 0.44
MAPK14 Q16539 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
PDE10A Q9Y233 1/20 0.40
PTGS2 P35354 2/20 0.40
KDM4E B2RXH2 1/20 0.39
CYP17A1 P05093 1/20 0.39
CYP1A2 P05177 1/20 0.39
KDM5A P29375 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
KDM5B Q9UGL1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27353154 0.83 POLB (0.53) MDM2NR3C2POLBMAPK9MAPK10
SCHEMBL1155787 0.80 MDM2 (0.55) MDM2NR3C2POLBMAPK9MAPK10
SCHEMBL27320127 0.79 MAPK9 (0.50) MDM2NR3C2POLBMAPK9MAPK10
SCHEMBL17086633 0.79 MDM2 (0.52) MDM2NR3C2POLBMAPK9MAPK10
SCHEMBL7067937 0.77 KDR (0.48) MDM2NR3C2POLBMAPK9MAPK10
SCHEMBL12759885 0.76 MDM2 (0.52) MDM2NR3C2MAPK9MAPK10MAPK8
SCHEMBL27323106 0.75 PDE10A (0.48) MDM2NR3C2POLBMAPK9MAPK10
SCHEMBL27315071 0.75 MAPK9 (0.68) MDM2NR3C2POLBMAPK9MAPK10
SCHEMBL27519346 0.75 NR3C2 (0.47) MDM2NR3C2POLBMAPK9MAPK10
SCHEMBL27730925 0.75 ALDH1A1 (0.55) MDM2NR3C2POLBMAPK9MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1031570-C Pyrazolopyridine compound and processes for preparation thereof FUJISAWA PHARMACEUTICAL CO (JP) 1996-04-17 CN disclosed
CN-1044656-A Pyrazolopyridine compound and preparation method thereof FUJISAWA PHARMACEUTICAL CO (JP) 1990-08-15 CN disclosed