SCHEMBL27360587

SCHEMBL27360587

Cc1cn([C@H](C(=O)N2CCC[C@H]2C(=O)N[C@@H](CO)c2ccc(-c3cnccc3C)cc2)C(C)C)cn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.35
PTGS2 P35354 1/20 0.35
ELANE P08246 3/20 0.34
XIAP P98170 1/20 0.34
MLX Q9UH92 1/20 0.34
ABL1 P00519 3/20 0.34
BRAF P15056 3/20 0.34
PREP P48147 1/20 0.33
FAP Q12884 1/20 0.33
MAPK1 P28482 2/20 0.33
VHL P40337 1/20 0.33
CCR5 P51681 1/20 0.33
KCNH2 Q12809 1/20 0.33
LRRK2 Q5S007 1/20 0.33
CCNK O75909 2/20 0.33
CDK12 Q9NYV4 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
FPR1 P21462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27360679 0.92 ROCK2 (0.37) ELANEXIAPMLXBRAFMAPK1
SCHEMBL27360586 0.91 DPP4 (0.40) ELANEXIAPMLXABL1BRAF
SCHEMBL27360684 0.87 CYP3A4 (0.34) ELANEXIAPMLXBRAFMAPK1
SCHEMBL27360583 0.86 DPP4 (0.37) ELANEXIAPMLXMAPK1KCNH2
SCHEMBL27360675 0.86 ELANE (0.38) ELANEXIAPMLXKCNH2CYP3A4
SCHEMBL27360670 0.85 ELANE (0.36) ELANEXIAPMLXMAPK1KCNH2
SCHEMBL27360584 0.85 ELANE (0.35) ELANEXIAPMLXMAPK1VHL
SCHEMBL27360367 0.78 XIAP (0.38) PTGESPTGS2ELANEXIAPMLX
SCHEMBL26847747 0.74 VHL (0.51) VHL
SCHEMBL27360361 0.72 MAPK1 (0.38) ELANEXIAPMLXPREPMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024040080-A1 KRAS INHIBITOR CONJUGATES ERASCA, INC. (US) 2024-02-22 WO disclosed