SCHEMBL27360583

SCHEMBL27360583

Cc1cn([C@H](C(=O)N2CCC[C@H]2C(=O)N[C@@H](CO)c2ccc(-c3ccccc3F)cc2)C(C)C)cn1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.37
TACR1 P25103 1/20 0.37
ELANE P08246 8/20 0.37
XIAP P98170 1/20 0.37
MLX Q9UH92 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KCNH2 Q12809 1/20 0.36
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
MAPK1 P28482 2/20 0.35
DPP7 Q9UHL4 2/20 0.34
PDE2A O00408 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
DPP8 Q6V1X1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27360584 0.94 ELANE (0.35) TACR1ELANEXIAPMLXCYP3A4
SCHEMBL27360670 0.91 ELANE (0.36) TACR1ELANEXIAPMLXCYP3A4
SCHEMBL27360675 0.89 ELANE (0.38) DPP4ELANEXIAPMLXCYP3A4
SCHEMBL27360679 0.88 ROCK2 (0.37) ELANEXIAPMLXKCNH2MAPK1
SCHEMBL27360587 0.86 PTGES (0.35) ELANEXIAPMLXCYP3A4CYP2C9
SCHEMBL27360684 0.85 CYP3A4 (0.34) ELANEXIAPMLXCYP3A4CYP2C9
SCHEMBL27360586 0.85 DPP4 (0.40) DPP4ELANEXIAPMLXKCNH2
SCHEMBL26847747 0.76 VHL (0.51)
SCHEMBL24756884 0.75 VHL (0.49)
SCHEMBL27360081 0.74 VHL (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024040080-A1 KRAS INHIBITOR CONJUGATES ERASCA, INC. (US) 2024-02-22 WO disclosed