SCHEMBL27369528

SCHEMBL27369528

Fc1cc(F)cc(F)c1.O=S(=O)(Cl)Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.43
CES1 P23141 3/20 0.43
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA9 Q16790 1/20 0.42
SOS1 Q07889 1/20 0.37
APLNR P35414 1/20 0.34
ACLY P53396 1/20 0.34
PTGS2 P35354 2/20 0.32
PTGS1 P23219 1/20 0.32
IDO1 P14902 2/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA13 Q8N1Q1 1/20 0.32
TGM2 P21980 1/20 0.31
PKM P14618 1/20 0.31
KMT2A Q03164 1/20 0.31
ALDH1A1 P00352 1/20 0.30
HSD17B10 Q99714 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5052222 0.86 CES2 (0.35) CES2CES1CA12CA1CA9
SCHEMBL67496 0.82 ALDH1A1 (0.42) CES2CES1CA12CA1CA9
SCHEMBL851628 0.82 CES2 (0.46) CES2CES1CA12CA1CA9
SCHEMBL28280990 0.80 PTGES2 (0.35) CES2CES1CA12CA1CA9
SCHEMBL28166420 0.79 CA1 (0.43) CES2CES1CA12CA1CA9
SCHEMBL1603078 0.79 CA1 (0.46) CES2CES1CA1CA9SOS1
SCHEMBL28282385 0.78 KDM1A (0.34) CES2CES1CA12CA1CA9
SCHEMBL3848319 0.78 CES2 (0.33) CES2CES1CA12CA1CA9
SCHEMBL9394710 0.76 IDO1 (0.38) CES2CES1CA12CA1CA9
SCHEMBL449836 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104045645-B The synthetic method of harringtonine C ring intermediates 河北科技大学 2018-10-19 CN claimed
CN-103265436-B Method for synthesising 1,5,9-trinitro-2,3,6,7,10,11-hexa-alkoxy triphenylene UNIV SHAANXI NORMAL 2015-03-18 CN claimed
CN-110325531-A Benzsulfamide and its purposes as therapeutic agent 泽农医药公司 2019-10-11 CN disclosed
CN-109526219-A Benzsulfamide and its purposes as therapeutic agent 泽农医药公司 2019-03-26 CN disclosed
CN-108698982-A FLUORINE ATOM-CONTAINING COMPOUND AND USE THEREOF 日产化学工业株式会社 2018-10-23 CN disclosed
CN-104045645-B The synthetic method of harringtonine C ring intermediates 河北科技大学 2018-10-19 CN disclosed
CN-105073114-B Medicine for respiratory disorder 第三共株式会社 2017-07-28 CN disclosed
CN-103265436-B Method for synthesising 1,5,9-trinitro-2,3,6,7,10,11-hexa-alkoxy triphenylene UNIV SHAANXI NORMAL 2015-03-18 CN disclosed
CN-104045646-A Synthetic method of harringtonine intermediate with D-ring UNIV HEBEI SCIENCE & TECH 2014-09-17 CN disclosed
CN-103265436-A Method for synthesising 1,5,9-trinitro-2,3,6,7,10,11-hexa-alkoxy triphenylene UNIV SHAANXI NORMAL 2013-08-28 CN disclosed
CN-101628888-B Inhibitors of cytosolic phospholipase a2 WYETH CORP 2012-05-23 CN disclosed
CN-101628888-A Inhibitors of cytosolic phospholipase A2 WYETH CORP 2010-01-20 CN disclosed
CN-100503566-C Cytosolic phospholipase A2 inhibitors WYETH CORP (US) 2009-06-24 CN disclosed
CN-1249039-C Inhibitors of 11 beta-hydroxysteroid dehydrogenase type I BIOVITRUM AB (SE) 2006-04-05 CN disclosed
CN-1617855-A Cytosolic phospholipase A2Inhibitors WYETH CORP (US) 2005-05-18 CN disclosed
CN-1438997-A Inhibitors of 11-beta-hydroxy steroid dehydrogenase type I BIOVITRUM AB (SE) 2003-08-27 CN disclosed
CN-1165144-A Phosphosulfonate herbicides ROHM & HAAS (US) 1997-11-19 CN disclosed
CN-1165143-A Phosphosulfonate herbicides ROHM & HAAS (US) 1997-11-19 CN disclosed
CN-1066266-A PHOSPHOSULFONATE HERBICIDES ROHM & HAAS (US) 1992-11-18 CN disclosed