Quinazolinone

Quinazolinone

SCHEMBL27369780

C1CCOC1.O=c1nc[nH]c2ccccc12

nearest known ligand 0.39

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.39
PDPK1 O15530 1/20 0.39
CA12 O43570 1/20 0.39
PARP1 P09874 1/20 0.39
ALOX15 P16050 1/20 0.39
CA9 Q16790 1/20 0.39
TNKS2 Q9H2K2 1/20 0.39
ALDH1A1 P00352 9/20 0.38
KMT2A Q03164 3/20 0.38
HPGD P15428 3/20 0.38
MAPT P10636 3/20 0.38
PRNP P04156 2/20 0.38
MEN1 O00255 2/20 0.38
HTT P42858 1/20 0.38
KDM4E B2RXH2 8/20 0.37
LMNA P02545 3/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
PDGFRB P09619 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinazolinone SCHEMBL10418 0.86 PARP1 (0.48) SMN1; SMN2PDPK1CA12PARP1ALOX15
Quinazolinone SCHEMBL7746268 0.84 PARP1 (0.47) SMN1; SMN2PDPK1CA12PARP1ALOX15
Quinazolinone SCHEMBL28241793 0.84 PARP1 (0.47) SMN1; SMN2PDPK1CA12PARP1ALOX15
Quinazolinone SCHEMBL8201415 0.84 PARP1 (0.47) SMN1; SMN2PDPK1CA12PARP1ALOX15
Quinazolinone SCHEMBL7744396 0.83 PARP1 (0.46) SMN1; SMN2PDPK1CA12PARP1ALOX15
Quinazolinone SCHEMBL27370560 0.77 PBRM1 (0.46) SMN1; SMN2PDPK1CA12PARP1ALOX15
Quinazolinone SCHEMBL27387957 0.77 PBRM1 (0.42) SMN1; SMN2PDPK1CA12PARP1ALOX15
Quinazolinone SCHEMBL5266556 0.75 ALDH1A1 (0.42) SMN1; SMN2PDPK1CA12PARP1ALOX15
Benzimidazole SCHEMBL28111344 0.75 KDM4E (0.41) SMN1; SMN2PDPK1CA12PARP1ALOX15
Benzimidazole SCHEMBL18329383 0.75 HPGD (0.40) SMN1; SMN2PDPK1CA12PARP1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1066847-A Angiotensin-ii receptor blockers 2,3,6 quinazolinones that replace AMERICAN CYANAMID CO (US) 1992-12-09 CN disclosed