Quinazolinone

Quinazolinone

SCHEMBL28241793

O=c1nc[nH]c2ccccc12.[H+]

nearest known ligand 0.47

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 8/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
PDPK1 O15530 1/20 0.47
CA12 O43570 1/20 0.47
ALOX15 P16050 1/20 0.47
CA9 Q16790 1/20 0.47
TNKS2 Q9H2K2 1/20 0.47
ALDH1A1 P00352 3/20 0.46
HPGD P15428 3/20 0.46
PRNP P04156 2/20 0.46
HTT P42858 2/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
KDM4E B2RXH2 3/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
ATM Q13315 2/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinazolinone SCHEMBL10418 0.98 PARP1 (0.48) PARP1SMN1; SMN2PDPK1CA12ALOX15
Quinazolinone SCHEMBL8201415 0.96 PARP1 (0.47) PARP1SMN1; SMN2PDPK1CA12ALOX15
Quinazolinone SCHEMBL7746268 0.96 PARP1 (0.47) PARP1SMN1; SMN2PDPK1CA12ALOX15
Quinazolinone SCHEMBL7744396 0.94 PARP1 (0.46) PARP1SMN1; SMN2PDPK1CA12ALOX15
Quinazolinone SCHEMBL27387957 0.87 PBRM1 (0.42) PARP1SMN1; SMN2PDPK1CA12ALOX15
Quinazolinone SCHEMBL27370560 0.87 PBRM1 (0.46) PARP1SMN1; SMN2PDPK1CA12ALOX15
Quinazolinone SCHEMBL5266556 0.86 ALDH1A1 (0.42) PARP1SMN1; SMN2PDPK1CA12ALOX15
Quinazolinone SCHEMBL27369780 0.84 SMN1; SMN2 (0.39) PARP1SMN1; SMN2PDPK1CA12ALOX15
Quinazolinone SCHEMBL28177707 0.78 CA12 (0.58) PARP1PDPK1CA12CA9CDK4
SCHEMBL29258736 0.75 PDE3B (0.44) PARP1SMN1; SMN2PDPK1CA12ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105189469-B 2-amino-3, 4-dihydroquinazoline derivatives and their use as cathepsin D inhibitors 默克专利股份公司 2018-09-25 CN disclosed
CN-106083741-A 2 sulfur are for quinazolinedione derivatives 南京中医药大学 2016-11-09 CN disclosed