SCHEMBL27382018

SCHEMBL27382018

Brc1cn(-c2cccc(N3CCN4CCC[C@H]4C3)c2)cn1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.47
POLB P06746 1/20 0.40
HTR6 P50406 4/20 0.39
ADCY5 O95622 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
HRH3 Q9Y5N1 2/20 0.39
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
MAP4K4 O95819 1/20 0.37
CTSS P25774 1/20 0.37
TSHR P16473 1/20 0.37
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38651777 1.00 HDAC4 (0.47) HDAC4POLBHTR6ADCY5HRH4
SCHEMBL38651646 0.88 HRH3 (0.46) HDAC4POLBHTR6HRH4HRH3
SCHEMBL27381924 0.80 FGFR1 (0.42) HDAC4POLBHTR6HRH3TSHR
SCHEMBL38651572 0.79 L3MBTL3 (0.46) HRH3
SCHEMBL38651513 0.79 L3MBTL3 (0.50) HRH3
SCHEMBL38651641 0.78 PIM1 (0.38) HTR6HRH4HRH3
SCHEMBL38651579 0.75 HTR6 (0.39) HTR6HRH4HRH3MAP4K4
SCHEMBL27380687 0.75 ADRA2C (0.50) HDAC4HRH4KMT2A
SCHEMBL38651750 0.75 ADRA2C (0.50) HDAC4HRH4KMT2A
SCHEMBL30773599 0.75 CTSS (0.41) HDAC4CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024062250-A1 IMIDAZOLYL-AMINO-PYRAZINE-CARBONITRILS AS CHK-1 INHIBITORS BENEVOLENTAI BIO LIMITED (GB) 2024-03-28 WO disclosed