SCHEMBL27405232

SCHEMBL27405232

CC(C(=O)O)c1cncnc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.45
HCAR2 Q8TDS4 1/20 0.44
PTGS1 P23219 10/20 0.42
AKR1C3 P42330 7/20 0.42
AKR1C2 P52895 6/20 0.42
CXCR1 P25024 4/20 0.42
CXCR2 P25025 4/20 0.42
LMNA P02545 3/20 0.42
SLC22A6 Q4U2R8 3/20 0.42
CYP2C9 P11712 2/20 0.42
CXCL8 P10145 2/20 0.42
PMP22 Q01453 2/20 0.42
TSHR P16473 2/20 0.42
ALB P02768 1/20 0.42
ESR1 P03372 1/20 0.42
ALOX5 P09917 1/20 0.42
RARB P10826 1/20 0.42
ADRB3 P13945 1/20 0.42
NFKB1 P19838 1/20 0.42
HTR2A P28223 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27922982 0.84 HCAR2 (0.41) HCAR2AKR1C3AKR1C2ALDH1A1
SCHEMBL1484347 0.80 EPHX1 (0.44) HCAR2
SCHEMBL1808417 0.80 HCAR2 (0.38) HCAR2
SCHEMBL1808418 0.77 HCAR2 (0.34) HCAR2
SCHEMBL26698325 0.75 HCAR2 (0.50) PTGS2HCAR2PTGS1AKR1C3AKR1C2
SCHEMBL29852325 0.75 HCAR2 (0.50) PTGS2HCAR2PTGS1AKR1C3AKR1C2
SCHEMBL6259017 0.75 AKR1C3 (0.57) PTGS2HCAR2PTGS1AKR1C3AKR1C2
SCHEMBL575045 0.75 AKR1C3 (0.57) PTGS2HCAR2PTGS1AKR1C3AKR1C2
SCHEMBL7446504 0.74 LMNA (0.50) HCAR2AKR1C3AKR1C2LMNATSHR
SCHEMBL30768172 0.74 PTGS2 (0.42) PTGS2PTGS1AKR1C3AKR1C2CXCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1085980-C Meta-guanidino, ureido, thioureido or azacyclic aminobenzoic acid derivatives as integrin antagonists SEARLE & CO (US) 2002-06-05 CN disclosed
CN-1201454-A Meta-guanidino, ureido, thioureido or azacyclic aminobenzoic acid derivatives as integrin antagonists SEARLE & CO (US) 1998-12-09 CN disclosed