SCHEMBL27411540

SCHEMBL27411540

N#Cc1cccnc1C(=O)c1cc(Cl)c(F)cc1O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.41
PDK2 Q15119 1/20 0.41
PDK3 Q15120 1/20 0.41
PDK4 Q16654 1/20 0.41
MALT1 Q9UDY8 1/20 0.40
CYP11B2 P19099 1/20 0.39
S1PR3 Q99500 8/20 0.39
S1PR1 P21453 4/20 0.39
GRM4 Q14833 2/20 0.39
GRM5 P41594 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.37
BACE1 P56817 1/20 0.35
AR P10275 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8713136 0.81 MEN1 (0.48) GRM5
SCHEMBL8714874 0.79 TLR7 (0.42) MALT1GRM4GRM5
SCHEMBL8712344 0.79 GRM4 (0.41) PDK1PDK2PDK3PDK4CYP11B2
SCHEMBL8709617 0.79 GRM4 (0.41) PDK1PDK2PDK3PDK4S1PR3
SCHEMBL8712498 0.78 PDK1 (0.35) PDK1PDK2PDK3PDK4MALT1
SCHEMBL8712738 0.77 KDM4C (0.40) GRM4GRM5
SCHEMBL27440948 0.76 HPGD (0.51)
SCHEMBL8715276 0.75 EGLN2 (0.39) PDK1PDK2PDK3PDK4GRM4
SCHEMBL8713994 0.74 P2RX7 (0.40) GRM4
SCHEMBL8709198 0.72 GRM4 (0.41) PDK1PDK2PDK3PDK4GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1097741-A Pyridine derivate, Preparation Method And The Use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-01-25 CN disclosed