SCHEMBL27412835

SCHEMBL27412835

Cc1ccc(C(=O)OC(=O)CC[C@H](N)C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 6/20 0.46
TDP1 Q9NUW8 1/20 0.42
SLC1A5 Q15758 2/20 0.41
GRIK1 P39086 2/20 0.41
GRIK2 Q13002 2/20 0.41
SLC1A1 P43005 2/20 0.41
GRM8 O00222 1/20 0.41
GRM6 O15303 1/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GSR P00390 1/20 0.41
CYP1A2 P05177 1/20 0.41
GRM5 P41594 1/20 0.41
GRIA1 P42261 1/20 0.41
GRIA2 P42262 1/20 0.41
GRIA3 P42263 1/20 0.41
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
GRIA4 P48058 1/20 0.41
GRIN1 Q05586 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1997087 0.86 SLC1A5 (0.48) KIF11SLC1A5GRIK1GRIK2SLC1A1
SCHEMBL9925277 0.86 SLC1A5 (0.48) KIF11SLC1A5GRIK1GRIK2SLC1A1
SCHEMBL6098839 0.81 TDP1 (0.57) TDP1NPC1RAB9AKMT2AALDH1A1
SCHEMBL9301762 0.77 SLC1A5 (0.49) KIF11TDP1SLC1A5NPC1RAB9A
Water SCHEMBL28445354 0.76 KMT2A (0.58) TDP1NPC1RAB9AKMT2AL3MBTL1
SCHEMBL8995839 0.76 TDP1 (0.52) TDP1CYP1A2NPC1RAB9AKMT2A
SCHEMBL5084403 0.76 ALDH1A1 (0.44) TDP1SLC1A5KMT2AL3MBTL1LTA4H
SCHEMBL5084405 0.76 ALDH1A1 (0.44) TDP1SLC1A5KMT2AL3MBTL1LTA4H
SCHEMBL28365251 0.75 TDP1 (0.47) TDP1NPC1RAB9AKMT2AALDH1A1
SCHEMBL5078447 0.75 LMNA (0.46) SLC1A5CYP1A2NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1394857-A Compound used as antiproliferative agent and glycinamide ribonucleotide transformylase inhibitor AQOURON PHARMACEUTICALS INC (US) 2003-02-05 CN disclosed
CN-1091770-C Compounds useful as antiproliferative agents and GARFT inhibitors AGOURON PHARAMCEUTICALS INC (US) 2002-10-02 CN disclosed
CN-1154110-A Compounds useful as antiproliferative agents and GARFT inhibitors AGOURON PHARMA (US) 1997-07-09 CN disclosed