SCHEMBL27422643

SCHEMBL27422643

ONNCc1ccc(Sc2ccc(CNNO)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.44
PTPRZ1 P23471 2/20 0.36
PTPN1 P18031 1/20 0.36
PTGIR P43119 1/20 0.35
THRB P10828 1/20 0.34
IDO1 P14902 1/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
MITF O75030 1/20 0.34
XBP1 P17861 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
NOD2 Q9HC29 1/20 0.34
HTT P42858 1/20 0.34
SLC6A4 P31645 3/20 0.33
CYP3A4 P08684 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549836 0.81 THRB (0.54) NR1H2PTPRZ1PTPN1PTGIRTHRB
SCHEMBL6540019 0.70 NR1H2 (0.52) NR1H2THRBMEN1KMT2AMAPT
SCHEMBL10887327 0.67 TSHR (0.48) NR1H2NPC1RAB9AMITFXBP1
SCHEMBL15826670 0.67 ESR1 (0.70) NR1H2PTPN1IDO1NPC1RAB9A
SCHEMBL6718210 0.67 ARG1 (0.57) NPSR1CYP1A2TSHRMAPK1MAPT
SCHEMBL14390455 0.64 NR1H2 (0.64) NR1H2IDO1SLC6A4CYP3A4MEN1
SCHEMBL588786 0.64 CA2 (0.56) NR1H2SLC6A4CYP3A4TSHRMAPK1
SCHEMBL10914949 0.63 NR1H2 (1.00) NR1H2THRBNPC1RAB9ACYP3A4
SCHEMBL29726 0.63 NR1H2 (1.00) NR1H2THRBNPC1RAB9ACYP3A4
SCHEMBL576175 0.62 TP53 (0.48) NR1H2IDO1SLC6A4CYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1045005-C Novel bisoxadiazolidine derivative YAMANOUCHI PHARMA CO LTD (JP) 1999-09-08 CN disclosed
CN-1122133-A Novel bis-oxadiazolidine derivatives YAMANOUCHI PHARMA CO LTD (JP) 1996-05-08 CN disclosed