SCHEMBL27424682

SCHEMBL27424682

CNc1ccnc(N2CCCc3ccccc32)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.57
ROCK1 Q13464 2/20 0.53
MAPT P10636 6/20 0.51
ALDH1A1 P00352 5/20 0.51
NPC1 O15118 4/20 0.51
RAB9A P51151 4/20 0.51
LMNA P02545 3/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
TP53 P04637 2/20 0.51
MAPK1 P28482 2/20 0.51
ALOX15 P16050 1/20 0.51
JAK2 O60674 1/20 0.46
JAK3 P52333 1/20 0.46
PTK2 Q05397 1/20 0.46
HPGD P15428 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5245431 0.80 ROCK1 (0.63) NUDT1ROCK1MAPTALDH1A1NPC1
SCHEMBL13911378 0.79 ROCK1 (0.56) NUDT1ROCK1MAPTALDH1A1NPC1
SCHEMBL5750076 0.76 ROCK1 (0.67) NUDT1ROCK1MAPTALDH1A1NPC1
SCHEMBL9004353 0.74 NUDT1 (0.51) NUDT1ROCK1MAPTALDH1A1NPC1
SCHEMBL2953620 0.73 HRH3 (0.51) ROCK1MAPTALDH1A1NPC1RAB9A
SCHEMBL13911376 0.72 ALDH1A1 (0.50) NUDT1ROCK1MAPTALDH1A1NPC1
SCHEMBL5414063 0.72 MAPT (0.57) NUDT1ROCK1MAPTALDH1A1NPC1
SCHEMBL19300445 0.71 ROCK1 (0.50) NUDT1ROCK1MAPTALDH1A1NPC1
SCHEMBL15831287 0.71 ROCK1 (0.55) ROCK1MAPTALDH1A1NPC1RAB9A
SCHEMBL10274926 0.70 ACHE (0.57) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1109675-C Aryl pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2003-05-28 CN disclosed
CN-1223641-A Aryl pyrimidine derivatives HOFFMANN LA ROCHE (CH) 1999-07-21 CN disclosed