SCHEMBL27425017

SCHEMBL27425017

CCC1CSc2ccc(-c3ccccc3)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 2/20 0.40
TMEM97 Q5BJF2 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
HTR1A P08908 1/20 0.40
DRD2 P14416 6/20 0.39
HTR2C P28335 1/20 0.35
FFAR1 O14842 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
DRD3 P35462 4/20 0.32
DRD4 P21917 3/20 0.32
HTR7 P34969 1/20 0.32
XIAP P98170 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13730382 0.64 DRD2 (0.39) HTR2BTMEM97SIGMAR1DRD2HTR2C
SCHEMBL21655317 0.61 KDM4C (0.43) MEN1NPC1USP2KMT2A
SCHEMBL25675893 0.61 KDM4C (0.43) MEN1NPC1USP2KMT2A
SCHEMBL9508981 0.59 ALDH1A1 (0.45) DRD2KDM4EMEN1NPC1USP2
SCHEMBL9511405 0.59 ALDH1A1 (0.45) DRD2KDM4EMEN1NPC1USP2
SCHEMBL21120521 0.59 DRD2 (0.35) DRD2KDM4EMEN1NPC1USP2
SCHEMBL24444333 0.59 MEN1 (0.44) HTR2BHTR2CKDM4EMEN1NPC1
Biphenyl SCHEMBL323849 0.59 ALDH1A1 (0.69) NPC1ALDH1A1MAPTHPGDSMN1; SMN2
Biphenyl SCHEMBL27803316 0.58 ALDH1A1 (0.50) ALDH1A1MAPTHPGDSMN1; SMN2
SCHEMBL24900236 0.58 MAOA (0.40) KDM4EMEN1USP2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1515567-A Novel benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake G.D.ɪ����˾ 2004-07-28 CN disclosed
CN-1110494-C Novel benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake SEARLE & CO (US) 2003-06-04 CN disclosed
CN-1221414-A Novel benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake SEARLE & CO (US) 1999-06-30 CN disclosed