SCHEMBL27428529

SCHEMBL27428529

CCC(=O)Oc1cnn(-c2ccnc(OCc3ccccc3)n2)c1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 6/20 0.39
KDM4C Q9H3R0 6/20 0.39
ALKBH1 Q13686 3/20 0.39
MAPK14 Q16539 2/20 0.37
KDM5B Q9UGL1 5/20 0.37
CYP1A2 P05177 4/20 0.37
ALDH1A1 P00352 4/20 0.36
TSHR P16473 3/20 0.36
CLK4 Q9HAZ1 1/20 0.36
MAPK1 P28482 2/20 0.35
LMNA P02545 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
HIF1A Q16665 1/20 0.35
PIK3CA P42336 1/20 0.35
FFAR1 O14842 1/20 0.34
KDM2B Q8NHM5 1/20 0.34
MAPK8 P45983 1/20 0.34
MAPK9 P45984 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7239669 0.80 NPC1 (0.49) CYP1A2ALDH1A1TSHRMAPK1LMNA
SCHEMBL27427760 0.79 TRPV1 (0.35) KDM5AKDM4CKDM5BALDH1A1HPGD
SCHEMBL27469144 0.79 HRH4 (0.48) KDM5AKDM4CALKBH1MAPK14CYP1A2
SCHEMBL27539537 0.73 VNN1 (0.42) ALDH1A1TSHRCLK4MAPK1
SCHEMBL27535631 0.72 KDM5A (0.46) KDM5AKDM4CKDM5BMAPK1HIF1A
SCHEMBL3804975 0.68 NPC1 (0.54) ALDH1A1MAPK1HPGD
SCHEMBL7229537 0.67 MAPK1 (0.50) KDM5AKDM4CALKBH1MAPK1CYP2C9
SCHEMBL18066391 0.66 FFAR4 (0.50) ALDH1A1MAPK1LMNACYP2C9CYP2C19
SCHEMBL28746011 0.65 LMNA (0.39) CYP1A2ALDH1A1TSHRLMNACYP2C19
SCHEMBL13403105 0.65 L3MBTL1 (0.47) KDM5AKDM4CCYP1A2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1105707-C Pyrazole derivative DAIICHI SEIYAKU CO (JP) 2003-04-16 CN disclosed
CN-1251578-A Pyrazole derivative DAIICHI SEIYAKU CO (JP) 2000-04-26 CN disclosed