Pyrilamine

Pyrilamine

SCHEMBL27430

COc1ccc(CN(CCN(C)C)c2ccccn2)cc1.O=C(O)/C=C\C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HRH1

The experimentally established mechanism targets of Pyrilamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 known ✓ P35367 5/20 0.80
SMN1; SMN2 Q16637 2/20 1.00
BLM P54132 1/20 1.00
PMP22 Q01453 1/20 1.00
LMNA P02545 4/20 0.80
CHRM2 P08172 3/20 0.80
ADRA2A P08913 3/20 0.80
DRD1 P21728 3/20 0.80
SLC6A4 P31645 3/20 0.80
SLC6A3 Q01959 3/20 0.80
KCNH2 Q12809 3/20 0.80
HTR2A P28223 2/20 0.80
CYP1A2 P05177 2/20 0.80
CYP2D6 P10635 2/20 0.80
TSHR P16473 2/20 0.80
CYP2C19 P33261 2/20 0.80
OPRM1 P35372 2/20 0.80
ALDH1A1 P00352 2/20 0.80
MEN1 O00255 1/20 0.80
CYP3A4 P08684 1/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyrilamine SCHEMBL2406435 1.00 SMN1; SMN2 (1.00) SMN1; SMN2BLMPMP22HRH1LMNA
Pyrilamine SCHEMBL97901 1.00 SMN1; SMN2 (1.00) SMN1; SMN2BLMPMP22HRH1LMNA
Pyrilamine SCHEMBL27517034 1.00 SMN1; SMN2 (1.00) SMN1; SMN2BLMPMP22HRH1LMNA
Pyrilamine SCHEMBL97902 1.00 SMN1; SMN2 (1.00) SMN1; SMN2BLMPMP22HRH1LMNA
Pyrilamine SCHEMBL5907722 0.99 SMN1; SMN2 (0.98) SMN1; SMN2BLMPMP22HRH1LMNA
Pyrilamine SCHEMBL11313804 0.92 SMN1; SMN2 (0.84) SMN1; SMN2BLMPMP22HRH1LMNA
Pyrilamine SCHEMBL9666725 0.91 SMN1; SMN2 (0.82) SMN1; SMN2BLMPMP22HRH1LMNA
Pyrilamine SCHEMBL9666718 0.91 SMN1; SMN2 (0.82) SMN1; SMN2BLMPMP22HRH1LMNA
Pyrilamine SCHEMBL4945522 0.90 SMN1; SMN2 (0.81) SMN1; SMN2BLMPMP22HRH1LMNA
Pyrilamine SCHEMBL622845 0.90 LMNA (0.95) SMN1; SMN2BLMPMP22HRH1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 31065 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250262177-A1 METHOD TO ALLEVIATE THE SYMPTOMS OF PMS CASH ALAN B (US) 2025-08-21 US claimed
EP-4149317-B1 CASE HOLOS PHARM SAGL (CH) 2024-07-17 EP claimed
EP-3152034-B1 MATERIAL PROCESSING METHODS AND RELATED APPARATUS HYBRID MANUFACTURING TECH LIMITED (GB) 2024-07-17 EP claimed
EP-3739138-B1 A PLAYGROUND KOMPAN AS (DK) 2024-07-10 EP claimed
EP-3503814-B1 INSTRUMENTATION FOR THE IMPLANTATION OF SPINAL IMPLANTS STRYKER EUROPEAN OPERATIONS HOLDINGS LLC (US) 2024-07-10 EP claimed
EP-3802215-B1 VEHICLE FOR TRANSPORTING GOODS FAYMONVILLE DISTRIB AG (LU) 2024-07-03 EP claimed
EP-4222373-B1 HOIST ARRANGEMENT FOR A WIND TURBINE BLADE ACCESS PLATFORM PP ENERGY APS (DK) 2024-07-03 EP claimed
EP-4393851-A1 LONG-LENGTH WOOD SORTING DEVICE Hans Hundegger Beteiligungs GmbH & Co. KG (DE) 2024-07-03 EP claimed
EP-4390117-A1 LIFTING MEANS FOR LIFTING A COMPONENT OF A WIND TURBINE Wobben Properties GmbH (DE) 2024-06-26 EP claimed
EP-4388925-A1 FIRST AID CASE, EMERGENCY CASE AND EMERGENCY CASE HALF, METHOD FOR CONNECTING TWO EMERGENCY CASE HALVES AND USE OF AN EMERGENCY CASE HALF W. Söhngen GmbH (DE) 2024-06-26 EP claimed
EP-0004858-A2 Bending apparatus for tubes L. ID. IT dei F.lli Belotti (IT) 1979-10-31 EP claimed
EP-0004282-A2 Hospital bed Joh. Stiegelmeyer & Co. GmbH (DE) 1979-10-03 EP claimed
WO-1979000682-A1 MACHINE FOR UNTYING AND REMOVING THE STRINGS AND BINDERS OF PACKED GOODS BORN AG P (CH) 1979-09-20 WO claimed
EP-0003998-A2 Machine for working a web of material by a welding tool STIEGLER GMBH MASCHINENFABRIK (DE) 1979-09-19 EP claimed
WO-1979000666-A1 MEASURING DEVICE FOR CHILLS IN CHILL-MOULDS FOR METAL,PARTICULARLY FOR STEEL SSAB SVENSKT STAL AB (SE) 1979-09-06 WO claimed
EP-0003574-A1 Method for positioning and supplying a stock of cups or closures, or longish tubular or bottle-like containers or the like to a filling machine Wiener Innovationsgesellschaft m.b.H. (AT) 1979-08-22 EP claimed
EP-0002188-A1 Treadmill for the therapy and rehabilitation of persons hampered in walking Schönenberger, Willi (CH) 1979-06-13 EP claimed
EP-0001967-A1 Apparatus for packing groups of articles in containers FOCKE & CO. (DE) 1979-05-30 EP claimed
EP-0001032-A1 Gas laser with transversal excitation ELTRO GmbH Gesellschaft für Strahlungstechnik (DE) 1979-03-07 EP claimed
EP-0000065-A1 Process and apparatus for bundling rods, tubes, profiles, and other oblong objects kabelmetal Messingwerke GmbH (DE) 1978-12-20 EP claimed