SCHEMBL27457403

SCHEMBL27457403

CC(=O)Nc1ccc(NS(=O)(=O)c2cc(C)c(S(=O)(=O)C[N+](=O)[O-])c(C)c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.58
MEN1 O00255 5/20 0.57
KMT2A Q03164 5/20 0.57
TDP1 Q9NUW8 2/20 0.57
KDM4E B2RXH2 1/20 0.57
CYP3A4 P08684 1/20 0.57
HPGD P15428 1/20 0.57
PKM P14618 2/20 0.55
GAA P10253 2/20 0.51
LMNA P02545 2/20 0.49
MAPK1 P28482 2/20 0.49
ALOX15 P16050 1/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
GFER P55789 1/20 0.49
KDM1A O60341 1/20 0.48
MAPT P10636 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7229750 0.93 PKM (0.62) ALDH1A1MEN1KMT2ATDP1KDM4E
SCHEMBL7226067 0.84 PKM (0.61) ALDH1A1MEN1KMT2ATDP1KDM4E
SCHEMBL7225299 0.84 ALDH1A1 (0.43) ALDH1A1MEN1KMT2ATDP1KDM4E
SCHEMBL9711178 0.81 KMT2A (0.60) ALDH1A1MEN1KMT2ATDP1KDM4E
SCHEMBL7224534 0.81 KMT2A (0.52) ALDH1A1MEN1KMT2ATDP1KDM4E
SCHEMBL7225029 0.78 ALDH1A1 (0.50) ALDH1A1MEN1KMT2ATDP1HPGD
SCHEMBL7221678 0.77 CYTH2 (0.56) ALDH1A1MEN1KMT2AHPGDPKM
SCHEMBL7221797 0.77 CYTH2 (0.43) ALDH1A1MEN1KMT2APKMGAA
SCHEMBL7223946 0.77 CYTH2 (0.46) ALDH1A1MEN1KMT2AHPGDPKM
SCHEMBL7222033 0.76 ALDH1A1 (0.39) ALDH1A1MEN1KMT2AKDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1112356-C Nitromethylthiobenzene derivatives as inhibitors of aldose reductase MERCK PATENT GMBH (DE) 2003-06-25 CN disclosed
CN-1241997-A Nitromethylthiobenzene derivatives as inhibitors of aldose reductase MERCK PATENT GMBH (DE) 2000-01-19 CN disclosed