SCHEMBL2747563

SCHEMBL2747563

CCc1ccccc1-c1cccc(S(=O)(=O)Nc2ccsc2C(=O)O)c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACLY P53396 5/20 0.52
NPSR1 Q6W5P4 1/20 0.45
PTGER3 P43115 1/20 0.45
IDH2 P48735 1/20 0.43
METAP2 P50579 1/20 0.43
NRP1 O14786 1/20 0.42
MCL1 Q07820 2/20 0.42
PFKFB3 Q16875 1/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2749453 0.90 LMNA (0.55) ACLYNPSR1PTGER3LMNAHPGD
SCHEMBL2748413 0.87 ACLY (0.54) ACLYNPSR1MCL1HPGDTSHR
SCHEMBL2748793 0.85 ACLY (0.62) ACLYNPSR1MCL1PFKFB3
SCHEMBL2748362 0.84 ACLY (0.51) ACLYNPSR1NRP1MCL1PFKFB3
SCHEMBL2747721 0.84 ACLY (0.47) ACLYNPSR1NRP1
SCHEMBL2747565 0.80 ACLY (0.56) ACLYNPSR1METAP2NRP1MCL1
SCHEMBL2747710 0.80 ACLY (0.59) ACLYNPSR1NRP1MCL1LMNA
SCHEMBL28646385 0.80 METAP2 (0.49) ACLYMETAP2MCL1PFKFB3LMNA
SCHEMBL532975 0.79 ACLY (0.69) ACLYNPSR1METAP2LMNAHPGD
Hydrochloric Acid SCHEMBL533067 0.77 ACLY (0.68) ACLYNPSR1METAP2LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178699-B2 Modulators of CCR9 receptor and methods of use thereof PFIZER INC. (US) 2012-05-15 US disclosed
US-8178699-B2 Modulators of CCR9 receptor and methods of use thereof PFIZER INC. (US) 2012-05-15 US disclosed
US-8178699-B2 Modulators of CCR9 receptor and methods of use thereof PFIZER INC. (US) 2012-05-15 US disclosed
EP-2220065-A2 MODULATORS OF CCR9 RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2010-08-25 EP disclosed
US-20100029753-A1 MODULATORS OF CCR9 RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. 2010-02-04 US disclosed
US-20100029753-A1 MODULATORS OF CCR9 RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. 2010-02-04 US disclosed
US-20100029753-A1 MODULATORS OF CCR9 RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. 2010-02-04 US disclosed
WO-2009017719-A2 MODULATORS OF CCR9 RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-02-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100029753-A1 MODULATORS OF CCR9 RECEPTOR AND METHODS OF USE THEREOF CCR9, CCR1, CCR4 ACLY 4546/4885NPSR1 220/4885PTGER3 705/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.