SCHEMBL28646385

SCHEMBL28646385

CCc1ccccc1-c1cccc(S(=O)(=O)Nc2cccc(C(=O)O)c2O)c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 2/20 0.49
PFKFB3 Q16875 1/20 0.48
KMT2A Q03164 6/20 0.48
MEN1 O00255 5/20 0.48
KDM4E B2RXH2 1/20 0.48
POLB P06746 1/20 0.48
MCL1 Q07820 4/20 0.47
GAA P10253 2/20 0.47
ACLY P53396 3/20 0.47
WDR5 P61964 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HSD17B10 Q99714 1/20 0.45
LMNA P02545 1/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28657757 0.91 METAP2 (0.52) METAP2PFKFB3KMT2AMEN1KDM4E
SCHEMBL28637411 0.88 ACLY (0.55) METAP2PFKFB3KMT2AMEN1KDM4E
SCHEMBL28926556 0.85 WDR5 (0.57) PFKFB3KMT2AMEN1KDM4EPOLB
SCHEMBL28925275 0.85 ACLY (0.49) PFKFB3KMT2AMEN1KDM4EPOLB
SCHEMBL28925257 0.84 MEN1 (0.52) PFKFB3KMT2AMEN1KDM4EPOLB
SCHEMBL28657550 0.84 MEN1 (0.50) PFKFB3KMT2AMEN1KDM4EPOLB
SCHEMBL28637197 0.84 MEN1 (0.50) PFKFB3KMT2AMEN1KDM4EPOLB
SCHEMBL28652663 0.84 PFKFB3 (0.55) PFKFB3KMT2AMEN1KDM4EPOLB
SCHEMBL28653065 0.82 PFKFB3 (0.48) PFKFB3KMT2AMEN1KDM4EPOLB
SCHEMBL2747563 0.80 ACLY (0.52) METAP2PFKFB3MCL1ACLYLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396145-A PFKFB3 inhibitors and uses thereof 盖罗发现有限责任公司 2021-09-14 CN disclosed