SCHEMBL27475645

SCHEMBL27475645

C=C(C(=O)N1CCN(C)CC1C(=O)OC)c1ccc(S)c(C(F)(F)F)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 2/20 0.34
PTK2 Q05397 3/20 0.33
LRRK2 Q5S007 1/20 0.33
MMP2 P08253 3/20 0.32
FKBP1A P62942 1/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
TAS1R2 Q8TE23 1/20 0.31
RBP4 P02753 1/20 0.31
TTR P02766 1/20 0.31
NOTUM Q6P988 1/20 0.31
EGFR P00533 1/20 0.31
SSTR4 P31391 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27490240 0.89 ALK (0.35) PDK2LRRK2MMP2FKBP1ANR1H2
SCHEMBL27492004 0.86 NR1H2 (0.40) NR1H2NR1H3
SCHEMBL6199381 0.79 ITGB2 (0.40)
SCHEMBL6197879 0.71 ITGB2 (0.45)
SCHEMBL27474903 0.70 SLC9A1 (0.45) HTR2ARBP4NOTUMSLC6A3
SCHEMBL6199011 0.70 ITGB2 (0.41)
SCHEMBL27490967 0.68 L3MBTL1 (0.43)
SCHEMBL7847221 0.68 HDAC4 (0.43) PDK2
SCHEMBL27475644 0.66 ITGAL (0.49) MMP2
SCHEMBL27475312 0.65 ITGB2 (0.42) MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1192018-C Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2005-03-09 CN claimed
CN-1353691-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2002-06-12 CN claimed
CN-1350520-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2002-05-22 CN claimed
CN-1955164-A Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds ABBOTT LAB (US) 2007-05-02 CN disclosed
CN-1680338-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2005-10-12 CN disclosed
CN-1192018-C Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2005-03-09 CN disclosed
CN-1353691-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2002-06-12 CN disclosed
CN-1350520-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2002-05-22 CN disclosed