SCHEMBL27490240

SCHEMBL27490240

C=C(C(=O)N1CCN(C(=O)OC)CC1C(=O)OC)c1ccc(S)c(C(F)(F)F)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.35
HSD11B1 P28845 1/20 0.34
PDK2 Q15119 2/20 0.33
MAPK3 P27361 1/20 0.33
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
LRRK2 Q5S007 4/20 0.33
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
TRPV4 Q9HBA0 1/20 0.32
EGFR P00533 1/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 2/20 0.32
PGR P06401 1/20 0.32
OPRK1 P41145 2/20 0.32
MMP2 P08253 2/20 0.31
FKBP1A P62942 1/20 0.31
TTK P33981 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27492004 0.93 NR1H2 (0.40) ALKNR1H2NR1H3MAPT
SCHEMBL27475645 0.89 PDK2 (0.34) PDK2NR1H2NR1H3LRRK2EGFR
SCHEMBL6199011 0.79 ITGB2 (0.41) MAPT
SCHEMBL6197045 0.76 ITGAL (0.35)
SCHEMBL6197879 0.75 ITGB2 (0.45)
SCHEMBL6197040 0.75 MEN1 (0.31) KMT2A
SCHEMBL27474903 0.74 SLC9A1 (0.45) ALKALDH1A1MAPTKMT2ACYP2C9
SCHEMBL27490967 0.74 L3MBTL1 (0.43) ALDH1A1MAPTKMT2ACYP2C19
SCHEMBL7847221 0.74 HDAC4 (0.43) PDK2ALDH1A1MAPTKMT2A
SCHEMBL6196692 0.72 ITGB2 (0.44) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1192018-C Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2005-03-09 CN claimed
CN-1353691-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2002-06-12 CN claimed
CN-1350520-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2002-05-22 CN claimed
CN-1955164-A Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds ABBOTT LAB (US) 2007-05-02 CN disclosed
CN-1680338-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2005-10-12 CN disclosed
CN-1192018-C Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2005-03-09 CN disclosed
CN-1353691-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2002-06-12 CN disclosed
CN-1350520-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2002-05-22 CN disclosed