SCHEMBL27475993

SCHEMBL27475993

COc1cc(OC)nc(N2CCNCC2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 4/20 0.56
HTR3E A5X5Y0 2/20 0.47
HTR3B O95264 2/20 0.47
HTR3A P46098 2/20 0.47
HTR3D Q70Z44 2/20 0.47
HTR3C Q8WXA8 2/20 0.47
CASP1 P29466 1/20 0.47
CASP4 P49662 1/20 0.47
CASP5 P51878 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
HTR1A P08908 1/20 0.47
HTR1D P28221 1/20 0.47
HTR1B P28222 1/20 0.47
HRH4 Q9H3N8 1/20 0.46
CHRNB2 P17787 1/20 0.44
CHRNA4 P43681 1/20 0.44
TGFBR1 P36897 1/20 0.44
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30124235 0.83 CASP1 (0.46) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2084347 0.81 CASP1 (0.47) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL27900639 0.77 HRH4 (0.43) ADRB1HRH4CHRNB2CHRNA4
SCHEMBL5988646 0.76 HTR2C (0.54) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL900166 0.76 ADRB1 (0.62) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL4430211 0.75 HTR2C (0.58) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2412819 0.75 HTR3E (0.58) ADRB1HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL11607113 0.74 HTR2C (0.57) ADRB1HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL3849292 0.74 HTR3E (0.57) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL14982162 0.74 ADRB1 (0.51) ADRB1HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1145609-C Piperazine compounds and medical use thereof ������ҩ��ʽ���� 2004-04-14 CN disclosed
CN-1281438-A Piperazine compounds and their use as pharmaceuticals EFUKU CO LTD (JP) 2001-01-24 CN disclosed