SCHEMBL27478043

SCHEMBL27478043

CC1=C(c2ccccc2)C=CC(C(=O)O)(c2nccn2C)C1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.35
ESR1 P03372 1/20 0.34
RIPK2 O43353 1/20 0.33
EGLN1 Q9GZT9 3/20 0.32
NTRK1 P04629 1/20 0.32
KMT2A Q03164 2/20 0.32
KDM4E B2RXH2 1/20 0.32
EGLN3 Q9H6Z9 1/20 0.31
OPRD1 P41143 2/20 0.30
FFAR1 O14842 1/20 0.30
CNR2 P34972 1/20 0.30
OPRK1 P41145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27494961 0.75
SCHEMBL27478874 0.73 RAB9A (0.37) KMT2AKDM4E
SCHEMBL27479658 0.71 KDM4E (0.33) KDM4E
SCHEMBL27478872 0.71 ALDH1A1 (0.35) KMT2AKDM4E
SCHEMBL27478044 0.71 NPC1 (0.35) KMT2AKDM4E
SCHEMBL30161783 0.70 KDM4E (0.33) KDM4E
SCHEMBL27529957 0.69 THRB (0.33)
SCHEMBL7922195 0.65 ADORA2A (0.37) NTRK1KDM4ECNR2
SCHEMBL27769281 0.65 ALOX5 (0.30)
SCHEMBL27968914 0.63 ALDH1A1 (0.33) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1175256-A tetracyclic spiro compounds, process for their preparation and their use as 5HT1D receptor antagonists SMITHKLINE BEECHAM PLC (GB) 1998-03-04 CN disclosed