SCHEMBL27485481

SCHEMBL27485481

O=C(O)/C=C/C1(c2ccccc2F)C=CC=NC1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
HDAC4 P56524 2/20 0.33
GAA P10253 1/20 0.33
ELOVL1 Q9BW60 1/20 0.31
LMNA P02545 1/20 0.30
BLM P54132 1/20 0.30
HCAR2 Q8TDS4 1/20 0.30
EGFR P00533 1/20 0.30
MMP1 P03956 1/20 0.30
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27502325 0.86 MEN1 (0.35) ALDH1A1LMNABLM
SCHEMBL27503047 0.85 CRHBP (0.35) HDAC4LMNABLMHDAC3HDAC1
SCHEMBL27561719 0.82 CDC25B (0.32) LMNA
SCHEMBL27484414 0.82 HCAR2 (0.33) HDAC4HCAR2HDAC3HDAC1HDAC2
SCHEMBL27484786 0.81 KDM4E (0.38)
SCHEMBL27529127 0.81 SLC6A2 (0.30)
SCHEMBL27486165 0.81 MAPT (0.42) ALDH1A1GAALMNA
SCHEMBL27504464 0.79 HSD11B1 (0.35) ALDH1A1GAALMNA
SCHEMBL27486162 0.75 CCR2 (0.34) ALDH1A1GAALMNA
SCHEMBL27504121 0.74 HSD11B1 (0.33) ALDH1A1HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1196721-A Heteroaryl-substituted acryloylguanidine derivatives and medicinal composition thereof YAMANOUCHI PHARMA CO LTD (JP) 1998-10-21 CN disclosed