SCHEMBL27489489

SCHEMBL27489489

O=CC(=O)c1cccc2cccnc12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.64
ALDH1A1 P00352 4/20 0.54
LMNA P02545 2/20 0.51
ALOX12 P18054 2/20 0.51
NPC1 O15118 3/20 0.50
CASP3 P42574 1/20 0.50
RAB9A P51151 1/20 0.50
SENP8 Q96LD8 1/20 0.50
SENP7 Q9BQF6 1/20 0.50
SENP6 Q9GZR1 1/20 0.50
MMP2 P08253 2/20 0.48
TSHR P16473 2/20 0.48
CHRM1 P11229 1/20 0.48
COMT P21964 1/20 0.48
ADRA1A P35348 1/20 0.48
METAP2 P50579 1/20 0.48
METAP1 P53582 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
TDP1 Q9NUW8 2/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27751301 0.84 PARP1 (0.62) PARP1ALDH1A1LMNAALOX12NPC1
SCHEMBL28050846 0.81 PARP1 (0.72) PARP1ALDH1A1LMNAALOX12NPC1
SCHEMBL9449256 0.80 PARP1 (0.57) PARP1ALDH1A1LMNAALOX12NPC1
SCHEMBL111826 0.79 PARP1 (0.70) PARP1ALDH1A1LMNAALOX12NPC1
SCHEMBL29749881 0.79 PARP1 (0.70) PARP1ALDH1A1LMNAALOX12NPC1
SCHEMBL27995395 0.79 MAPT (0.49) PARP1ALDH1A1LMNAALOX12NPC1
SCHEMBL16859274 0.78 PARP1 (0.68) PARP1ALDH1A1LMNAALOX12NPC1
SCHEMBL1164312 0.78 PARP1 (0.68) PARP1ALDH1A1LMNAALOX12NPC1
SCHEMBL4507521 0.78 PARP1 (0.68) PARP1ALDH1A1LMNAALOX12NPC1
Hydrochloric Acid SCHEMBL7320778 0.78 PARP1 (0.68) PARP1ALDH1A1LMNAALOX12NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108299415-B Quinolinequinone derivative and preparation method and application thereof 南通大学 2020-11-10 CN claimed
CN-108299415-A A kind of quinoline quinone derivative and preparation method and purposes 南通大学 2018-07-20 CN claimed
CN-100519533-C 5-arylamino quinolyl-7,8-dione derivative and its application in preparing antibiotic medicine UNIV GUANGDONG TECHNOLOGY (CN) 2009-07-29 CN claimed
CN-1974557-A 5-arylamino quinolyl-7,8-dione derivative and its application in preparing antibiotic medicine UNIV GUANGDONG POLYTECHNIC (CN) 2007-06-06 CN claimed
CN-113214149-B Synthesis method of phenyl (quinoline-8-yl) ketone derivative 江苏师范大学 2022-08-02 CN disclosed
CN-113214149-A Synthesis method of phenyl (quinoline-8-yl) ketone derivative 江苏师范大学 2021-08-06 CN disclosed
CN-108299415-B Quinolinequinone derivative and preparation method and application thereof 南通大学 2020-11-10 CN disclosed
CN-110218198-A A kind of naphthoquinones and triazole core skeleton derivative compound and its preparation method and application 广州中医药大学(广州中医药研究院) 2019-09-10 CN disclosed
CN-109020986-A Quinoline quinone and oxa- ring derivatives and preparation method thereof and the application on anti-tumor drug 中南大学 2018-12-18 CN disclosed
CN-108299415-A A kind of quinoline quinone derivative and preparation method and purposes 南通大学 2018-07-20 CN disclosed
CN-100374438-C Pre-organized tricyclic integrase inhibitor compounds GILEAD SCIENCES INC (US) 2008-03-12 CN disclosed
CN-1726212-A Pre-organized tricyclic integrase inhibitor compounds GILEAD SCIENCES INC (US) 2006-01-25 CN disclosed
CN-1187352-C Phenanthroline-7-one derivatives and their therapeutic use LAFON LABOR (FR) 2005-02-02 CN disclosed
CN-1139575-C Process for preparing quinoline-5, 8-diones L���������鹫˾ 2004-02-25 CN disclosed
CN-1129582-C 3-substituted-4-arylquinolin-2-one derivatives as potassium channel modulators BRISTOL MYERS SQUIBB CO (US) 2003-12-03 CN disclosed
CN-1373761-A Phenanthroline-7-one derivatives and their therapeutic use LAFON LABOR (FR) 2002-10-09 CN disclosed
CN-1370149-A Process for preparing quinoline-5, 8-diones LAFON LABOR (FR) 2002-09-18 CN disclosed
CN-1344269-A Pharmaceutical compsn. based on polyaromatic compounds LAFON LABOR (FR) 2002-04-10 CN disclosed
CN-1329599-A 3-substituted-4-arylquinolin-2-one derivatives as potassium channel modulators BRISTOL MYERS SQUIBB CO (US) 2002-01-02 CN disclosed