SCHEMBL9449256

SCHEMBL9449256

[N-]=[N+]=CC(=O)c1cccc2cccnc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.57
ALDH1A1 P00352 4/20 0.49
ALOX12 P18054 2/20 0.47
LMNA P02545 2/20 0.47
NPC1 O15118 4/20 0.46
RAB9A P51151 2/20 0.46
CASP3 P42574 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
MMP2 P08253 2/20 0.43
TSHR P16473 2/20 0.43
CHRM1 P11229 1/20 0.43
COMT P21964 1/20 0.43
ADRA1A P35348 1/20 0.43
METAP2 P50579 1/20 0.43
METAP1 P53582 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
KDM4E B2RXH2 5/20 0.43
MAPT P10636 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27489489 0.80 PARP1 (0.64) PARP1ALDH1A1ALOX12LMNANPC1
SCHEMBL27751301 0.79 PARP1 (0.62) PARP1ALDH1A1ALOX12LMNANPC1
SCHEMBL6642077 0.78 P2RX7 (0.50) ALDH1A1LMNANPC1RAB9ATSHR
SCHEMBL28050846 0.76 PARP1 (0.72) PARP1ALDH1A1ALOX12LMNANPC1
SCHEMBL111826 0.74 PARP1 (0.70) PARP1ALDH1A1ALOX12LMNANPC1
SCHEMBL29749881 0.74 PARP1 (0.70) PARP1ALDH1A1ALOX12LMNANPC1
SCHEMBL8801910 0.74 ALDH1A1 (0.41) ALDH1A1LMNATSHRKDM4EMAPT
SCHEMBL8978021 0.73 NR4A1 (0.53) ALDH1A1LMNANPC1RAB9ATSHR
SCHEMBL29883614 0.73 NR4A1 (0.53) ALDH1A1LMNANPC1RAB9ATSHR
SCHEMBL2632726 0.73 PARP1 (0.68) PARP1ALDH1A1ALOX12LMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0466730-B1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1993-07-21 EP disclosed
US-5220021-A Geminal bisphosphonic acids and derivatives as anti-arthritic agents THE UPJOHN COMPANY (US) 1993-06-15 US disclosed
WO-1990012017-A1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1990-10-18 WO disclosed