SCHEMBL27499151

SCHEMBL27499151

CN(C)Cc1cc(CC(C)(C)OC(N)=O)c([N+](=O)[O-])cc1I

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.33
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP2C19 P33261 2/20 0.31
ALOX15 P16050 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
ALDH1A1 P00352 1/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27484337 0.87 PARP1 (0.35) PARP1CYP2C19ALOX15HTTALDH1A1
SCHEMBL27539422 0.85 HCAR3 (0.38) PARP1MAPTSMN1; SMN2MAPK1HTT
SCHEMBL27500363 0.83 PDGFRB (0.38) PARP1MAPTSMN1; SMN2CYP2C19ALOX15
SCHEMBL27520362 0.83 SNCA (0.40) PARP1MAPTSMN1; SMN2CYP2C19ALOX15
SCHEMBL27554338 0.83 ALDH1A1 (0.36) PARP1ALDH1A1
SCHEMBL27499148 0.82 CTSD (0.36) PARP1MAPTCYP2C19HTTALDH1A1
SCHEMBL27486075 0.81 ALDH1A1 (0.46) PARP1MAPTSMN1; SMN2ALDH1A1
SCHEMBL27498854 0.81 ALDH1A1 (0.35) PARP1SMN1; SMN2CYP2C19HTTALDH1A1
SCHEMBL27485132 0.77 PARP1 (0.37) PARP1SMN1; SMN2CYP2C19HTTALDH1A1
SCHEMBL28742589 0.77 HCAR3 (0.39) MAPTSMN1; SMN2MAPK1HTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1195522-C Benzodiazepine derivatives usable as parental metabolic glutamate receptor antagonist HOFFMANN LA ROCHE (CH) 2005-04-06 CN disclosed
CN-1379765-A Benzodiazepine derivatives usable as parental metabolic glutamate receptor antagonist HOFFMANN LA ROCHE (CH) 2002-11-13 CN disclosed