SCHEMBL27554338

SCHEMBL27554338

CC(C)(Cc1cc(CC#N)c(I)cc1[N+](=O)[O-])OC(N)=O

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27484337 0.86 PARP1 (0.35) ALDH1A1PARP1
SCHEMBL27499151 0.83 PARP1 (0.33) ALDH1A1PARP1
SCHEMBL27520362 0.82 SNCA (0.40) ALDH1A1PARP1
SCHEMBL27500363 0.82 PDGFRB (0.38) ALDH1A1PARP1
SCHEMBL27499148 0.81 CTSD (0.36) ALDH1A1HPGDPARP1
SCHEMBL27498854 0.80 ALDH1A1 (0.35) ALDH1A1PARP1
SCHEMBL27539422 0.80 HCAR3 (0.38) ALDH1A1HPGDPARP1
SCHEMBL27485132 0.76 PARP1 (0.37) ALDH1A1PARP1
SCHEMBL27485057 0.76 MAPT (0.37) ALDH1A1
SCHEMBL27486073 0.75 BACE1 (0.41) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1195522-C Benzodiazepine derivatives usable as parental metabolic glutamate receptor antagonist HOFFMANN LA ROCHE (CH) 2005-04-06 CN disclosed
CN-1379765-A Benzodiazepine derivatives usable as parental metabolic glutamate receptor antagonist HOFFMANN LA ROCHE (CH) 2002-11-13 CN disclosed