SCHEMBL27505437

SCHEMBL27505437

COC(=O)CC(N)CC(C)Cc1cccc(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A1 P43005 2/20 0.47
SLC7A5 Q01650 2/20 0.45
DPP4 P27487 2/20 0.43
DPP7 Q9UHL4 2/20 0.43
MAOB P27338 3/20 0.41
MAOA P21397 2/20 0.41
ROCK1 Q13464 1/20 0.41
SCN9A Q15858 1/20 0.41
ROCK2 O75116 1/20 0.40
ANPEP P15144 1/20 0.40
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
FAP Q12884 1/20 0.39
DPP8 Q6V1X1 1/20 0.39
DPP9 Q86TI2 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27489377 0.85 PNMT (0.52) SLC7A5DPP4DPP7MAOBDPP8
SCHEMBL27488012 0.84 HTT (0.43) DPP4DPP7TSHR
SCHEMBL27488009 0.84 MMP1 (0.49) SLC7A5MAOAANPEP
SCHEMBL4332275 0.80 SLC1A1 (0.48) SLC1A1DPP4DPP7ROCK1
Hydrochloric Acid SCHEMBL4326709 0.79 SLC1A1 (0.47) SLC1A1DPP4DPP7ROCK1
SCHEMBL27507829 0.77 DPP4 (0.41) DPP4DPP7SCN9APPARGPPARA
SCHEMBL27488015 0.77 SLC1A1 (0.43) SLC1A1SLC7A5MAOBMAOASCN9A
SCHEMBL27506206 0.76 SLC6A2 (0.46) DPP4DPP7CYP2D6CYP2C9CYP2C19
SCHEMBL27505438 0.75 SLC1A1 (0.57) SLC1A1SLC7A5DPP4DPP7ROCK1
SCHEMBL75362 0.74 SLC1A1 (0.55) SLC1A1SLC7A5DPP4DPP7MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101862317-A The pregabalin derivant that is used for the treatment of fibromyalgia and other disease WARNER LAMBERT CO 2010-10-20 CN disclosed
CN-1310872-C Mono- and disubstituted 3-propyl gamma-aminobutyric acids WARNER LAMBERT CO (US) 2007-04-18 CN disclosed
CN-1726023-A Pregabalin derivatives for the treatment of fibromyalgia and other diseases WARNER LAMBERT CO (US) 2006-01-25 CN disclosed
CN-1660779-A Mono- and disubstituted 3-propyl gamma-aminobutyric acids WARNER LAMBERT CO (US) 2005-08-31 CN disclosed
CN-1625393-A Alpha 2 delta ligands to treat tinnitus WARNER LAMBERT CO (US) 2005-06-08 CN disclosed
CN-1196671-C Mono-and disubstituted 3-propyl-gamma-aminobutyric acids WARNER LAMBERT CO (US) 2005-04-13 CN disclosed
CN-1355784-A Mono-and disubstituted 3-propyl-gamma-aminobutyric acids WARNER LAMBERT CO (US) 2002-06-26 CN disclosed