SCHEMBL27488012

SCHEMBL27488012

COC(=O)CC(N)CC(C)Cc1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.40
TRPA1 O75762 1/20 0.40
CA12 O43570 3/20 0.39
CA7 P43166 3/20 0.39
CA9 Q16790 3/20 0.39
CA14 Q9ULX7 3/20 0.39
CA2 P00918 1/20 0.39
DPP4 P27487 1/20 0.39
DPP7 Q9UHL4 1/20 0.39
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GAA P10253 1/20 0.39
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27506206 0.86 SLC6A2 (0.46) DPP4DPP7KMT2AGAA
SCHEMBL27488009 0.86 MMP1 (0.49) MEN1KMT2AMMP1
SCHEMBL28200415 0.85 HTT (0.49) HTTALDH1A1MAPTHPGDTSHR
SCHEMBL27505437 0.84 SLC1A1 (0.47) TSHRDPP4DPP7
SCHEMBL27507829 0.78 DPP4 (0.41) ALDH1A1DPP4DPP7KMT2ATDP1
SCHEMBL23551731 0.77 TSHR (0.50) HTTHPGDTSHRTRPA1CA12
SCHEMBL27489377 0.76 PNMT (0.52) ALDH1A1HPGDDPP4DPP7KMT2A
SCHEMBL20134406 0.74 TSHR (0.48) HTTHPGDTSHRTRPA1CA12
SCHEMBL8283148 0.74 TSHR (0.48) HTTHPGDTSHRTRPA1CA12
SCHEMBL27506588 0.74 CA12 (0.47) HTTALDH1A1MAPTHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101862317-A The pregabalin derivant that is used for the treatment of fibromyalgia and other disease WARNER LAMBERT CO 2010-10-20 CN disclosed
CN-1310872-C Mono- and disubstituted 3-propyl gamma-aminobutyric acids WARNER LAMBERT CO (US) 2007-04-18 CN disclosed
CN-1726023-A Pregabalin derivatives for the treatment of fibromyalgia and other diseases WARNER LAMBERT CO (US) 2006-01-25 CN disclosed
CN-1660779-A Mono- and disubstituted 3-propyl gamma-aminobutyric acids WARNER LAMBERT CO (US) 2005-08-31 CN disclosed
CN-1625393-A Alpha 2 delta ligands to treat tinnitus WARNER LAMBERT CO (US) 2005-06-08 CN disclosed
CN-1196671-C Mono-and disubstituted 3-propyl-gamma-aminobutyric acids WARNER LAMBERT CO (US) 2005-04-13 CN disclosed
CN-1355784-A Mono-and disubstituted 3-propyl-gamma-aminobutyric acids WARNER LAMBERT CO (US) 2002-06-26 CN disclosed