Dalfampridine

Dalfampridine

SCHEMBL27520243

Nc1ccncc1.O=CO

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2

The experimentally established mechanism targets of Dalfampridine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA1 known ✓ Q09470 1/20 0.68
MAPT P10636 6/20 0.68
ALDH1A1 P00352 3/20 0.68
MEN1 O00255 3/20 0.68
KMT2A Q03164 3/20 0.68
CYP2D6 P10635 2/20 0.68
LMNA P02545 2/20 0.68
CHRM1 P11229 1/20 0.68
TSHR P16473 1/20 0.68
MAPK1 P28482 1/20 0.68
SMN1; SMN2 Q16637 1/20 0.68
RAD52 P43351 1/20 0.44
CYP3A4 P08684 2/20 0.40
CYP19A1 P11511 2/20 0.40
CYP17A1 P05093 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
POLB P06746 1/20 0.39
NAPRT Q6XQN6 1/20 0.39
KDM4E B2RXH2 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dalfampridine SCHEMBL28027907 0.89 MAPT (0.77) MAPTALDH1A1MEN1KMT2ACYP2D6
Dalfampridine SCHEMBL53483 0.83
Dalfampridine SCHEMBL1442620 0.83 MAPT (1.00) MAPTALDH1A1MEN1KMT2ACYP2D6
Dalfampridine SCHEMBL27592753 0.81 MAPT (0.72) MAPTALDH1A1MEN1KMT2ACYP2D6
Dalfampridine SCHEMBL28737546 0.80
Dalfampridine SCHEMBL7987482 0.80
Dalfampridine SCHEMBL7113651 0.80
Dalfampridine SCHEMBL28629661 0.80
Dalfampridine SCHEMBL28750367 0.80 MAPT (0.93) MAPTALDH1A1MEN1KMT2ACYP2D6
Dalfampridine SCHEMBL3845825 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 52 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105072897-B Temperature stabilization cloquitocet_mexyl Aquo-composition 美国陶氏益农公司 2017-04-05 CN claimed
CN-105072897-A Temperature stable cloquintocet-mexyl aqueous compositions DOW AGROSCIENCES LLC 2015-11-18 CN claimed
CN-104994734-A SYNERGISTIC WEED CONTROL FROM APPLICATIONS OF AMINOPYRALID AND CLOPYRALID DOW AGROSCIENCES LLC 2015-10-21 CN claimed
CN-102605356-B Plating catalyst and method ROHM & HAAS ELECT MAT 2014-11-19 CN claimed
CN-1281591-C 4-aminopyridinecarboxylates and their use as herbicides DOW AGROSCIENCES LLC (US) 2006-10-25 CN claimed
CN-110461819-A Process for the preparation of benzyl 4-amino-3-chloro-5-fluoro-6- (4-chloro-2-fluoro-3-methoxyphenyl) picolinate DOW AGROSCIENCES LLC 2019-11-15 CN disclosed
CN-106279012-B A kind of preparation method of 3,4,6- trichloropyridine -2- formic acid and its ester 利尔化学股份有限公司 2019-04-09 CN disclosed
CN-106459060-B Condensed triazole derivative as phosphodiesterase 10 A inhibitor 赛隆制药股份公司 2019-04-05 CN disclosed
CN-104994734-B Collaboration control of weeds is carried out by application chloroaminopyridine acid and clopyralid 美国陶氏益农公司 2018-06-29 CN disclosed
CN-108135157-A Complexes of cloquintocet-mexyl and amine-containing polymers or oligomers 美国陶氏益农公司 2018-06-08 CN disclosed
CN-104994735-B Using the collaboration control of weeds caused by the pyrimidine acid of ring third and 2,4 dichlorophenoxyacetic acids (2,4 drop) 美国陶氏益农公司 2017-12-12 CN disclosed
CN-104988531-B The method that a kind of selective dechlorination of chloro-pyridine formic acid electro-catalysis prepares pyridine carboxylic acid 浙江工业大学 2017-11-07 CN disclosed
CN-1823045-A 6-(1,1-difluoroalkyl)-4-aminopicolinates and their use as herbicides DOW AGROSCIENCES LLC (US) 2006-08-23 CN disclosed
CN-1764646-A 6-alkyl-or alkenyl-4-aminopicolinates and their use as herbicides DOW AGROSCIENCES LLC (US) 2006-04-26 CN disclosed
CN-1751042-A Pyrazolo[3,4-b]pyridine compounds, and their use as phosphodiesterase inhibitors GLAXO GROUP LTD (GB) 2006-03-22 CN disclosed
CN-1245401-C 6-aryl-4-aminopicolinates and their use as herbicides DOW AGROSCIENCES LLC (US) 2006-03-15 CN disclosed
CN-1238565-C Selective electrochemical reduction of halogenated 4-aminopicolinic acids DOW AGROSCIENCES LLC (US) 2006-01-25 CN disclosed
CN-1551876-A 6-aryl-4-aminopicolinates and their use as herbicides �ݶ�ũ�����޹�˾ 2004-12-01 CN disclosed
CN-1416419-A 4-aminopyridinecarboxylates and their use as herbicides DOW AGROSCIENCES LLC (US) 2003-05-07 CN disclosed
CN-1394241-A Selective electrochemical reduction of halogenated 4-aminopicolinic acids DOW AGROSCIENCES LLC (US) 2003-01-29 CN disclosed