SCHEMBL27535652

SCHEMBL27535652

COc1ccc(C(C(C)=O)c2ccc(O)cc2)c(O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYR P14679 2/20 0.49
BCHE P06276 1/20 0.49
ACHE P22303 1/20 0.49
CYP3A4 P08684 3/20 0.49
HPGD P15428 2/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPK1 P28482 1/20 0.49
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
PPARG P37231 1/20 0.46
KMT2A Q03164 1/20 0.46
TRIM24 O15164 1/20 0.41
TRIM33 Q9UPN9 1/20 0.41
PTGS2 P35354 3/20 0.41
AKR1C3 P42330 3/20 0.41
AKR1C2 P52895 3/20 0.41
PTGS1 P23219 2/20 0.41
CYP1A2 P05177 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16836085 0.85 TYR (0.46) TYRCYP3A4ALDH1A1MEN1MAPT
SCHEMBL4443109 0.82 CYP3A4 (0.56) TYRBCHEACHECYP3A4HPGD
SCHEMBL8153518 0.80 MAOB (0.44) TYRBCHEACHECYP3A4MEN1
SCHEMBL11558507 0.79 HPGD (0.50) TYRBCHEACHECYP3A4HPGD
SCHEMBL16685610 0.78 TUBB4A (0.43) TYRBCHEACHECYP3A4ALDH1A1
SCHEMBL4656144 0.78 BCHE (0.54) TYRBCHEACHECYP3A4NPC1
SCHEMBL9391336 0.76 CES2 (0.50) NPC1RAB9AMEN1MAPTKMT2A
SCHEMBL4731187 0.76 TYR (0.49) TYRBCHEACHECYP3A4HPGD
SCHEMBL5144377 0.75 ESR1 (0.55) TYRBCHEACHECYP3A4HPGD
SCHEMBL788027 0.75 LMNA (0.44) CYP3A4HPGDALDH1A1MAPK1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1281598-C Compounds and methods for modulation of estrogen receptors SIGNAL PHARM INC (US) 2006-10-25 CN disclosed
CN-1437591-A Compounds and methods for modulation of estrogen receptors SIGNAL PHARM INC (US) 2003-08-20 CN disclosed