SCHEMBL27536722

SCHEMBL27536722

CNc1ccc(C(C)C(=O)C(C)c2ccc(NC)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
RECQL P46063 2/20 0.42
HSD17B10 Q99714 2/20 0.42
HPGD P15428 2/20 0.42
TP53 P04637 1/20 0.42
CYP3A4 P08684 1/20 0.42
THRB P10828 1/20 0.42
ALOX15 P16050 1/20 0.42
CASP1 P29466 1/20 0.42
HIF1A Q16665 1/20 0.42
PTGS2 P35354 4/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
NR1H4 Q96RI1 1/20 0.39
FFAR2 O15552 1/20 0.39
KIF11 P52732 1/20 0.39
CHRM1 P11229 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL693789 0.85 PTGS2 (0.57) ALDH1A1HPGDPTGS2NR1H4PTGS1
SCHEMBL10760564 0.83 EPHX1 (0.55) ALDH1A1RECQLHSD17B10HPGDTP53
SCHEMBL14386006 0.83 EPHX1 (0.55) ALDH1A1RECQLHSD17B10HPGDTP53
SCHEMBL11272564 0.82 HPGD (0.49) ALDH1A1RECQLHSD17B10HPGDTP53
SCHEMBL27536587 0.81 RXFP1 (0.50) ALDH1A1RECQLHSD17B10CYP3A4THRB
SCHEMBL27536643 0.78 MAPT (0.43) HPGDPTGS2SMN1; SMN2GAAMAPT
SCHEMBL11586901 0.77 LMNA (0.47) HPGDPTGS2SMN1; SMN2CA12CA1
SCHEMBL27512331 0.77 CYP2C9 (0.48) ALDH1A1HPGDHIF1APTGS2SMN1; SMN2
SCHEMBL28003757 0.76 LMNA (0.58) ALDH1A1RECQLHPGDSMN1; SMN2KIF11
SCHEMBL28806262 0.75 MEN1 (0.46) MEN1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1252070-A 5,7-disubstituted 4-aminopyrido [2,3,-d] pyrimidine compounds and their use as adenosine kinase inhibitors ABBOTT LAB (US) 2000-05-03 CN disclosed