Trazodone

Trazodone

SCHEMBL27570399

CCO.O=c1n(CCCN2CCN(c3cccc(Cl)c3)CC2)nc2ccccn12

nearest known ligand 0.90

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HTR2AHTR2CSLC6A4

The experimentally established mechanism targets of Trazodone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A known ✓ P28223 11/20 0.90
HTR2C known ✓ P28335 3/20 0.90
SLC6A4 known ✓ P31645 3/20 0.90
DRD2 P14416 11/20 0.90
HTR1A P08908 10/20 0.90
ADRA2A P08913 3/20 0.90
ADRA2B P18089 3/20 0.90
ADRA2C P18825 3/20 0.90
DRD1 P21728 3/20 0.90
DRD4 P21917 3/20 0.90
ADRA1A P35348 3/20 0.90
HRH1 P35367 3/20 0.90
DRD3 P35462 3/20 0.90
KDM4E B2RXH2 2/20 0.90
ALDH1A1 P00352 2/20 0.90
HPGD P15428 2/20 0.90
HSD17B10 Q99714 2/20 0.90
ABCB11 O95342 2/20 0.90
HRH2 P25021 2/20 0.90
TACR1 P25103 2/20 0.90

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trazodone SCHEMBL28167 0.95 HTR1A (1.00) DRD2HTR2AHTR1AADRA2AADRA2B
Trazodone SCHEMBL29390760 0.95 HTR1A (1.00) DRD2HTR2AHTR1AADRA2AADRA2B
Trazodone SCHEMBL28226073 0.94 HTR1A (0.98) DRD2HTR2AHTR1AADRA2AADRA2B
Trazodone SCHEMBL29575935 0.94 KDM4E (1.00) DRD2HTR2AHTR1AADRA2AADRA2B
Trazodone SCHEMBL3402550 0.94 KDM4E (1.00) DRD2HTR2AHTR1AADRA2AADRA2B
Trazodone SCHEMBL61754 0.94 KDM4E (1.00) DRD2HTR2AHTR1AADRA2AADRA2B
Trazodone SCHEMBL8741340 0.93 DRD2 (0.89) DRD2HTR2AHTR1AADRA2AADRA2B
Trazodone SCHEMBL120883 0.93 HTR1A (0.96) DRD2HTR2AHTR1AADRA2AADRA2B
SCHEMBL11089944 0.93 HTR1A (0.98) DRD2HTR2AHTR1AADRA2AADRA2B
Trazodone SCHEMBL23145121 0.91 HTR1A (0.87) DRD2HTR2AHTR1AADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1341852-A Quick testing method of rape erucidic and reagent INST OF OIL CROPS CHINESE ACAD (CN) 2002-03-27 CN disclosed