SCHEMBL27587441

SCHEMBL27587441

O=C(O)CC[C@H](F)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.48
ALDH1A1 P00352 2/20 0.48
CYP2C19 P33261 2/20 0.48
CYP1A2 P05177 1/20 0.48
TSHR P16473 1/20 0.48
CPA3 P15088 1/20 0.47
NAALAD2 Q9Y3Q0 1/20 0.46
KEAP1 Q14145 1/20 0.43
MAPK1 P28482 3/20 0.42
KDM4E B2RXH2 1/20 0.42
TP53 P04637 1/20 0.42
GLA P06280 1/20 0.42
POLB P06746 1/20 0.42
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
ALOX12 P18054 1/20 0.42
NFKB1 P19838 1/20 0.42
APEX1 P27695 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NR4A2 P43354 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27985511 1.00 CYP2D6 (0.48) CYP2D6ALDH1A1CYP2C19CYP1A2TSHR
SCHEMBL4063595 1.00 CYP2D6 (0.48) CYP2D6ALDH1A1CYP2C19CYP1A2TSHR
SCHEMBL11822261 0.89 FFAR1 (0.50) CYP2D6ALDH1A1CYP2C19CYP1A2TSHR
SCHEMBL27587412 0.88 HDAC3 (0.47) CYP2D6ALDH1A1CYP2C19CYP1A2TSHR
SCHEMBL7319044 0.86 TBXAS1 (0.53) CYP2D6ALDH1A1CYP2C19CYP1A2TSHR
SCHEMBL23757780 0.84 ALDH1A1 (0.47) CYP2D6ALDH1A1CYP2C19CYP1A2TSHR
SCHEMBL3674189 0.80 CYP2D6 (0.54) CYP2D6ALDH1A1CYP2C19CYP1A2TSHR
SCHEMBL23570862 0.80 CA12 (0.48) ALDH1A1TSHRKDM4EPOLBHSD17B10
SCHEMBL16426389 0.80 CA12 (0.48) ALDH1A1TSHRKDM4EPOLBHSD17B10
SCHEMBL7390419 0.78 GABBR2 (0.53) CYP2D6CYP2C19CPA3MAPK1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104159595-A Peptidomimetic macrocycles AILERON THERAPEUTICS INC 2014-11-19 CN disclosed
CN-104144695-A Triazole-and thioether-crosslinked peptidomimetic macrocycles AILERON THERAPEUTICS INC 2014-11-12 CN disclosed
CN-104039342-A Peptidomimetic macrocycles AILERON THERAPEUTICS INC 2014-09-10 CN disclosed
CN-1512983-A Compounds and compositions as cathepsins inhibitors AXYSҩ�﹫˾ 2004-07-14 CN disclosed