SCHEMBL27587795

SCHEMBL27587795

CC(=O)Nc1ccc(-c2c(C#N)c(N)[nH]c(=S)c2C#N)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.59
MAPT P10636 5/20 0.59
KDM4E B2RXH2 3/20 0.59
ALOX15 P16050 1/20 0.59
HSD17B10 Q99714 1/20 0.59
ADORA3 P0DMS8 1/20 0.53
ADORA2A P29274 1/20 0.53
ADORA2B P29275 1/20 0.53
PFKFB1 P16118 1/20 0.50
UBE2N P61088 1/20 0.49
GAA P10253 3/20 0.46
CUL4A Q13619 1/20 0.45
HTT P42858 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
RXFP1 Q9HBX9 2/20 0.42
PPARG P37231 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27572255 0.88 MAPT (0.46) ALDH1A1MAPTKDM4EALOX15HSD17B10
SCHEMBL935141 0.75 ALDH1A1 (1.00) ALDH1A1MAPTKDM4EALOX15HSD17B10
SCHEMBL3064294 0.75 MAPT (0.67) ALDH1A1MAPTKDM4EALOX15HSD17B10
SCHEMBL7013023 0.73 ADORA3 (0.65) ALDH1A1MAPTKDM4EALOX15HSD17B10
SCHEMBL19720089 0.73 PFKFB1 (0.50) ALDH1A1MAPTKDM4EADORA3ADORA2A
SCHEMBL4306407 0.72 ADORA3 (0.64) ALDH1A1MAPTKDM4EALOX15HSD17B10
SCHEMBL23885077 0.70 PFKFB1 (0.76) ALDH1A1KDM4EALOX15HSD17B10PFKFB1
SCHEMBL30052633 0.70 PFKFB1 (0.76) ALDH1A1KDM4EALOX15HSD17B10PFKFB1
SCHEMBL8472800 0.69 SMN1; SMN2 (0.50) ALDH1A1MAPTKDM4EADORA3ADORA2A
SCHEMBL1778210 0.69 KDM4E (0.58) ALDH1A1MAPTKDM4EALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1407971-A Substituted 2-thio-3,5-dicyano-4-aryl-6-aminopyridines and the use thereof BAYER AG (DE) 2003-04-02 CN disclosed